SCHEMBL3821500

SCHEMBL3821500

N#Cc1ccc(N(Cc2ccccc2C(F)(F)F)C2CCN(C(=O)CN)C2)cc1Cl

nearest known ligand 0.85

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PGR P06401 20/20 0.85
CYP2D6 P10635 17/20 0.85
CYP2C9 P11712 17/20 0.85
AR P10275 2/20 0.71
KCNH2 Q12809 2/20 0.71
NR3C1 P04150 1/20 0.71
NR3C2 P08235 1/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3821495 1.00 PGR (0.85) PGRCYP2D6CYP2C9ARKCNH2
SCHEMBL3862670 0.91 PGR (0.83) PGRCYP2D6CYP2C9ARKCNH2
SCHEMBL14162317 0.91 PGR (0.83) PGRCYP2D6CYP2C9ARKCNH2
SCHEMBL3862673 0.91 PGR (0.83) PGRCYP2D6CYP2C9ARKCNH2
SCHEMBL3025306 0.91 PGR (0.85) PGRCYP2D6CYP2C9ARKCNH2
SCHEMBL14162228 0.90 PGR (0.81) PGRCYP2D6CYP2C9ARKCNH2
SCHEMBL14162266 0.88 PGR (0.66) PGRCYP2D6CYP2C9ARKCNH2
SCHEMBL3828660 0.87 PGR (1.00) PGRCYP2D6CYP2C9ARKCNH2
SCHEMBL3828666 0.87 PGR (1.00) PGRCYP2D6CYP2C9ARKCNH2
SCHEMBL14162319 0.87 PGR (0.86) PGRCYP2D6CYP2C9ARKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2094269-A1 PYRROLIDINANILINES Smithkline Beecham Corporation (US) 2009-09-02 EP disclosed
WO-2008077089-A1 PYRROLIDINANILINES SMITHKLINE BEECHAM CORPORATION (US) 2008-06-26 WO disclosed