SCHEMBL3821840

SCHEMBL3821840

[NH]C1CCN(c2ccc(Cl)c(C(F)(F)F)n2)CC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACACB O00763 2/20 0.44
ADRB2 P07550 1/20 0.43
HTR3E A5X5Y0 1/20 0.37
MEN1 O00255 1/20 0.37
HTR3B O95264 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
ALOX15 P16050 1/20 0.37
TSHR P16473 1/20 0.37
NFKB1 P19838 1/20 0.37
HTR3A P46098 1/20 0.37
KMT2A Q03164 1/20 0.37
HTR3D Q70Z44 1/20 0.37
HTR3C Q8WXA8 1/20 0.37
HRH3 Q9Y5N1 3/20 0.36
RXFP1 Q9HBX9 1/20 0.35
KDM4E B2RXH2 2/20 0.34
MAPT P10636 2/20 0.34
ABL1 P00519 1/20 0.34
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18908932 0.85 ACACB (0.47) ACACBADRB2HTR3EMEN1HTR3B
SCHEMBL3821841 0.85 HTR3E (0.54) ACACBADRB2HTR3EMEN1HTR3B
SCHEMBL23762505 0.83 ACACB (0.45) ACACBADRB2HTR3EMEN1HTR3B
SCHEMBL4504026 0.80 ACACB (0.48) ACACBHTR3EMEN1HTR3BCYP1A2
SCHEMBL4504023 0.80 ACACB (0.48) ACACBHTR3EMEN1HTR3BCYP1A2
SCHEMBL30455678 0.73 ACACB (0.40) ACACB
SCHEMBL18176137 0.68 CYP1A2 (0.38) ACACBADRB2CYP1A2TSHRLMNA
SCHEMBL28544593 0.67 ACACB (0.33) ACACBADRB2
SCHEMBL23404890 0.65 ACACB (0.34) ACACB
SCHEMBL23405058 0.65 ACACB (0.38) ACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009143018-A2 COMPOUNDS AND METHODS FOR KINASE MODULATION, AND INDICATIONS THEREFOR PLEXXIKON, INC. (US) 2009-11-26 WO disclosed
EP-1603899-B1 HETEROCYCLIC UREA DERIVATIVES FOR THE TREATMENT OF PAIN GLAXO GROUP LTD (GB) 2009-08-26 EP disclosed