SCHEMBL3822220

SCHEMBL3822220

N#Cc1ccc(N(CC2CCCC2)[C@H]2CCN(C(=O)O)C2)cc1Cl

nearest known ligand 0.71

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PGR P06401 20/20 0.71
CYP2C9 P11712 16/20 0.59
CYP2D6 P10635 15/20 0.59
KCNH2 Q12809 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14162419 0.89 PGR (0.69) PGRCYP2C9CYP2D6KCNH2
SCHEMBL14162365 0.87 PGR (0.71) PGRCYP2C9CYP2D6KCNH2
SCHEMBL3819111 0.87 PGR (0.71) PGRCYP2C9CYP2D6KCNH2
SCHEMBL3819105 0.87 PGR (0.71) PGRCYP2C9CYP2D6KCNH2
SCHEMBL3821469 0.86 PGR (0.66) PGRCYP2C9CYP2D6KCNH2
SCHEMBL14162183 0.86 PGR (0.69) PGRCYP2C9CYP2D6KCNH2
SCHEMBL3821463 0.86 PGR (0.66) PGRCYP2C9CYP2D6KCNH2
SCHEMBL14162418 0.86 PGR (0.69) PGRCYP2C9CYP2D6KCNH2
SCHEMBL14162407 0.86 PGR (0.69) PGRCYP2C9CYP2D6KCNH2
SCHEMBL14162429 0.86 PGR (0.63) PGRCYP2C9CYP2D6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2094269-A1 PYRROLIDINANILINES Smithkline Beecham Corporation (US) 2009-09-02 EP disclosed
WO-2008077089-A1 PYRROLIDINANILINES SMITHKLINE BEECHAM CORPORATION (US) 2008-06-26 WO disclosed