SCHEMBL3822277

SCHEMBL3822277

COc1cc(COC(=O)c2ccc3c(c2)CCC(C)(C)O3)cc(OC)c1OC

nearest known ligand 0.68

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
COXFA4 O00483 2/20 0.68
HSP90AA1 P07900 3/20 0.54
HTT P42858 2/20 0.45
PDE7A Q13946 3/20 0.44
PDE3A Q14432 3/20 0.44
PDE4B Q07343 1/20 0.44
PDE4D Q08499 1/20 0.44
PDE7B Q9NP56 1/20 0.44
OPRM1 P35372 1/20 0.44
PDE10A Q9Y233 1/20 0.43
MGAM O43451 3/20 0.41
GAA P10253 3/20 0.41
SI P14410 3/20 0.41
MGAM2 Q2M2H8 3/20 0.41
MAPT P10636 2/20 0.41
LMNA P02545 1/20 0.41
ALDH1A1 P00352 1/20 0.41
TSHR P16473 1/20 0.41
GHSR Q92847 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3456476 0.85 COXFA4 (0.77) COXFA4HSP90AA1HTTOPRM1PDE10A
SCHEMBL3456261 0.81 COXFA4 (0.61) COXFA4HSP90AA1HTTPDE7APDE3A
SCHEMBL14139260 0.81 COXFA4 (1.00) COXFA4HSP90AA1HTTOPRM1PDE10A
SCHEMBL31026771 0.80 COXFA4 (0.50) COXFA4MGAMGAASIMGAM2
SCHEMBL6210404 0.80 COXFA4 (0.50) COXFA4MGAMGAASIMGAM2
SCHEMBL12315569 0.80 COXFA4 (0.59) COXFA4HSP90AA1HTTPDE7APDE3A
SCHEMBL16742142 0.78 COXFA4 (0.53) COXFA4MGAMGAASIMGAM2
SCHEMBL12677576 0.78 COXFA4 (0.72) COXFA4HSP90AA1PDE4BPDE4DOPRM1
SCHEMBL12315585 0.78 COXFA4 (0.60) COXFA4HSP90AA1PDE4DOPRM1PDE10A
SCHEMBL9850284 0.78 HIF1A (0.49) COXFA4MGAMGAASIMGAM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1740225-A4 CONTRAST AGENTS FOR MYOCARDIAL PERFUSION IMAGING BRISTOL MYERS SQUIBB CO (US) 2009-08-19 EP disclosed
US-7410998-B2 Inhibitors of NADH:ubiquinone oxidoreductase THE SCRIPPS RESEARCH INSTITUTE (US) 2008-08-12 US disclosed
EP-1740225-A2 CONTRAST AGENTS FOR MYOCARDIAL PERFUSION IMAGING Bristol-Myers Squibb Company (US) 2007-01-10 EP disclosed
WO-2005105159-A2 CONTRAST AGENTS FOR MYOCARDIAL PERFUSION IMAGING BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2005-11-10 WO disclosed