SCHEMBL3825923

SCHEMBL3825923

[NH]C(=O)C1CN1C(c1ccccc1)(c1ccccc1)c1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 4/20 0.36
CHRM2 P08172 3/20 0.36
CHRM1 P11229 3/20 0.36
KEAP1 Q14145 1/20 0.35
NFE2L2 Q16236 1/20 0.35
CYP1A2 P05177 1/20 0.34
ALDH1A1 P00352 1/20 0.33
CHRM4 P08173 1/20 0.33
CHRM5 P08912 1/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.32
KMT2A Q03164 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4047414 0.85 CHRM2 (0.38) CHRM3CHRM2CHRM1KEAP1NFE2L2
SCHEMBL23274047 0.85 CHRM2 (0.38) CHRM3CHRM2CHRM1KEAP1NFE2L2
SCHEMBL991996 0.85 CHRM2 (0.38) CHRM3CHRM2CHRM1KEAP1NFE2L2
SCHEMBL23415467 0.84 CHRM2 (0.37) CHRM3CHRM2CHRM1KEAP1NFE2L2
SCHEMBL23415469 0.84 CHRM2 (0.37) CHRM3CHRM2CHRM1KEAP1NFE2L2
SCHEMBL23415565 0.84 CHRM2 (0.37) CHRM3CHRM2CHRM1KEAP1NFE2L2
SCHEMBL3825928 0.82 MAPT (0.40) CHRM3CHRM2CHRM1KEAP1NFE2L2
SCHEMBL25897057 0.82 CHRM3 (0.36) CHRM3CHRM2CHRM1KEAP1NFE2L2
Lithium Ion SCHEMBL29888438 0.81 CHRM3 (0.35) CHRM3CHRM2CHRM1KEAP1NFE2L2
SCHEMBL30537611 0.81 CHRM3 (0.35) CHRM3CHRM2CHRM1KEAP1NFE2L2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2099747-A1 RADIOLABELLING VIA FLUORINATION OF AZIRIDINES Bayer Schering Pharma Aktiengesellschaft (DE) 2009-09-16 EP disclosed
WO-2008083729-A1 RADIOLABELLING VIA FLUORINATION OF AZIRIDINES BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2008-07-17 WO disclosed
EP-1944288-A1 Radiolabelling via fluorination of aziridines Bayer Schering Pharma Aktiengesellschaft (DE) 2008-07-16 EP disclosed