SCHEMBL3826352

SCHEMBL3826352

O=C1CC=CN=C1C#Cc1ccc(N2CCC(Oc3ccccc3F)CC2)nc1

nearest known ligand 0.43

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
RET P07949 1/20 0.39
DCK P27707 6/20 0.39
SCD O00767 1/20 0.36
GPR6 P46095 2/20 0.36
GRM5 P41594 2/20 0.35
SCN9A Q15858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3831479 0.79 GRM5 (0.45) RETDCKSCDGRM5
SCHEMBL3847667 0.77 DCK (0.46) RETDCKSCD
SCHEMBL14130746 0.77 RET (0.44) RETDCKSCDGPR6
SCHEMBL3828744 0.74 DCK (0.46) RETDCKSCD
SCHEMBL3826351 0.72 RET (0.42) RETDCKGPR6GRM5SCN9A
SCHEMBL3832548 0.72 RET (0.42) RETDCKGPR6GRM5SCN9A
SCHEMBL14143777 0.68 SCD (0.52) RETDCKSCDGPR6
SCHEMBL3831437 0.68 CYP3A4 (0.42) SCD
SCHEMBL3854486 0.67 CYP3A4 (0.41) SCD
SCHEMBL3826490 0.67 SCD (0.46) DCKSCDGPR6SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2099755-A2 ACETYLENE DERIVATIVES AS STEAROYL COA DESATURASE INHIBITORS Glenmark Pharmaceuticals S.A. (CH) 2009-09-16 EP disclosed
WO-2008062276-A2 ACETYLENE DERIVATIVES AS STEAROYL COA DESATURASE INHIBITORS GLENMARK PHARMACEUTICALS S.A. (US) 2008-05-29 WO disclosed