SCHEMBL3828302

SCHEMBL3828302

CCCN1C[N]c2ccccc21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
ALDH1A1 P00352 2/20 0.44
MAPT P10636 2/20 0.39
KDM4E B2RXH2 1/20 0.39
NSD2 O96028 1/20 0.39
ADRA2A P08913 2/20 0.38
ADRA2B P18089 2/20 0.38
ADRA2C P18825 2/20 0.38
LMNA P02545 1/20 0.37
NISCH Q9Y2I1 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C19 P33261 1/20 0.36
DRD2 P14416 3/20 0.35
THRB P10828 1/20 0.35
ATM Q13315 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
ALOX12 P18054 1/20 0.34
TAAR1 Q96RJ0 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7345950 0.82 ALDH1A1 (0.49) MEN1KMT2AALDH1A1MAPTKDM4E
SCHEMBL7351385 0.80 ALDH1A1 (0.54) MEN1KMT2AALDH1A1MAPTKDM4E
SCHEMBL21834896 0.76 MEN1 (0.52) MEN1KMT2AALDH1A1MAPTKDM4E
SCHEMBL28252759 0.75 MEN1 (0.41) MEN1KMT2AALDH1A1MAPTKDM4E
SCHEMBL5540573 0.74 ALDH1A1 (0.34) ALDH1A1MAPTKDM4ENSD2ADRA2C
SCHEMBL7345538 0.73 CYP2D6 (0.43) MEN1KMT2AALDH1A1KDM4ELMNA
SCHEMBL6196442 0.71 MEN1 (0.45) MEN1KMT2AALDH1A1KDM4ELMNA
SCHEMBL3697070 0.71 ALDH1A1 (0.47) MEN1KMT2AALDH1A1MAPTKDM4E
SCHEMBL9330383 0.71 MEN1 (0.47) MEN1KMT2AALDH1A1MAPTADRA2A
SCHEMBL7352919 0.70 POLB (0.37) MEN1KMT2AALDH1A1MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1414825-B9 THIENOPYRIMIDINEDIONES AND THEIR USE IN THE MODULATION OF AUTOIMMUNE DISEASE ASTRAZENECA AB (SE) 2009-09-16 EP disclosed
EP-1414825-B1 THIENOPYRIMIDINEDIONES AND THEIR USE IN THE MODULATION OF AUTOIMMUNE DISEASE ASTRAZENECA AB (SE) 2007-09-26 EP disclosed