SCHEMBL3829055

SCHEMBL3829055

CC1(CN(C(=O)O)C(C)(C)C)CCN(Cc2ccccc2)C1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 7/20 0.46
CYP3A4 P08684 2/20 0.46
TSHR P16473 2/20 0.46
OPRM1 P35372 2/20 0.42
SIGMAR1 Q99720 1/20 0.42
GAA P10253 1/20 0.42
CHRM2 P08172 1/20 0.41
CHRM3 P20309 1/20 0.41
ALDH1A1 P00352 2/20 0.41
DRD2 P14416 1/20 0.41
DRD4 P21917 1/20 0.41
DRD3 P35462 1/20 0.41
OPRL1 P41146 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14716322 0.93 CYP2D6 (0.50) CYP2D6CYP3A4TSHROPRM1SIGMAR1
SCHEMBL1313447 0.82 CYP2D6 (0.50) CYP2D6CYP3A4TSHROPRM1SIGMAR1
SCHEMBL16684766 0.76 OPRL1 (0.51) CYP2D6CYP3A4TSHRSIGMAR1GAA
SCHEMBL28282362 0.76 CYP2D6 (0.51) CYP2D6CYP3A4TSHROPRM1GAA
SCHEMBL6603001 0.75 OPRM1 (0.47) CYP2D6TSHROPRM1SIGMAR1ALDH1A1
SCHEMBL3272594 0.74 CYP2D6 (0.49) CYP2D6CYP3A4TSHRGAACHRM2
SCHEMBL12596337 0.74 CYP3A4 (0.51) CYP2D6CYP3A4TSHRSIGMAR1GAA
SCHEMBL14342254 0.74 NPFFR1 (0.48) CYP2D6CYP3A4TSHRALDH1A1
SCHEMBL12372531 0.73 CYP2D6 (0.51) CYP2D6CYP3A4TSHROPRM1GAA
SCHEMBL27926426 0.73 CYP2D6 (0.47) CYP2D6CYP3A4TSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1796466-A4 ANTIBACTERIAL AGENTS GLAXO GROUP LTD (GB) 2009-09-02 EP disclosed
EP-1796466-A2 ANTIBACTERIAL AGENTS GLAXO GROUP LIMITED (GB) 2007-06-20 EP disclosed
WO-2006002047-A2 ANTIBACTERIAL AGENTS GLAXO GROUP LIMITED (GB) 2006-01-05 WO disclosed