SCHEMBL3835582

SCHEMBL3835582

CC(C)(O)C(=O)N1CCC(N(Cc2ccccc2F)c2ccc(C#N)c(Cl)c2)C1

nearest known ligand 0.79

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PGR P06401 20/20 0.79
CYP2C9 P11712 19/20 0.79
CYP2D6 P10635 17/20 0.79
KCNH2 Q12809 2/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3835584 1.00 PGR (0.79) PGRCYP2C9CYP2D6KCNH2
SCHEMBL14162236 0.93 PGR (0.79) PGRCYP2C9CYP2D6KCNH2
SCHEMBL3821530 0.91 PGR (0.68) PGRCYP2C9CYP2D6KCNH2
SCHEMBL3821528 0.91 PGR (0.68) PGRCYP2C9CYP2D6KCNH2
SCHEMBL14162316 0.90 PGR (0.66) PGRCYP2C9CYP2D6KCNH2
SCHEMBL3824734 0.89 PGR (0.83) PGRCYP2C9CYP2D6KCNH2
SCHEMBL14162245 0.89 PGR (0.83) PGRCYP2C9CYP2D6KCNH2
SCHEMBL3821428 0.88 PGR (0.77) PGRCYP2C9CYP2D6KCNH2
SCHEMBL3821421 0.88 PGR (0.77) PGRCYP2C9CYP2D6KCNH2
SCHEMBL3826305 0.87 PGR (0.81) PGRCYP2C9CYP2D6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2094269-A1 PYRROLIDINANILINES Smithkline Beecham Corporation (US) 2009-09-02 EP claimed
WO-2008077089-A1 PYRROLIDINANILINES SMITHKLINE BEECHAM CORPORATION (US) 2008-06-26 WO claimed
EP-2094269-A1 PYRROLIDINANILINES Smithkline Beecham Corporation (US) 2009-09-02 EP disclosed
WO-2008077089-A1 PYRROLIDINANILINES SMITHKLINE BEECHAM CORPORATION (US) 2008-06-26 WO disclosed