SCHEMBL3835849

SCHEMBL3835849

CCCOc1cc2c(c(-c3cc4cc(CN5CCN(CCO)CC5)ccc4n3C(=O)OC(C)(C)C)c1)C(=O)NC2

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 11/20 0.39
ALDH1A1 P00352 1/20 0.38
MEN1 O00255 1/20 0.37
NPC1 O15118 1/20 0.37
TP53 P04637 1/20 0.37
GAA P10253 1/20 0.37
RAB9A P51151 1/20 0.37
KMT2A Q03164 1/20 0.37
AURKA O14965 1/20 0.35
KDR P35968 1/20 0.35
PKM P14618 1/20 0.34
ATR Q13535 2/20 0.34
ATRIP Q8WXE1 2/20 0.34
GPR4 P46093 1/20 0.33
NR1H3 Q13133 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3863205 0.92 HRH3 (0.39) NR1H2AURKAKDRNR1H3
SCHEMBL3837061 0.89 NTRK1 (0.36) NR1H2PKMATRATRIPNR1H3
SCHEMBL3855204 0.85 ALDH1A1 (0.35) NR1H2ALDH1A1MEN1NPC1TP53
SCHEMBL3839112 0.85 NR1H2 (0.38) NR1H2NR1H3
SCHEMBL3834957 0.83 ATR (0.38) NR1H2ATRATRIPNR1H3
SCHEMBL3859943 0.82 NR1H2 (0.35) NR1H2ATRATRIPNR1H3
SCHEMBL3840220 0.82 ATR (0.35) NR1H2AURKAKDRATRATRIP
SCHEMBL3166857 0.82 NR1H2 (0.37) NR1H2ALDH1A1KDRPKMATR
SCHEMBL3043824 0.82 NR1H2 (0.38) NR1H2ALDH1A1GAAKDRPKM
SCHEMBL3835632 0.81 PARP1 (0.40) NR1H2NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2108642-A1 JAK INHIBITOR Kyowa Hakko Kirin Co., Ltd. (JP) 2009-10-14 EP disclosed