SCHEMBL3836682

SCHEMBL3836682

O=C(N[C@H]1CC[C@@](O)(C#Cc2cccc(Cl)c2)CC1)Oc1ccccn1

nearest known ligand 0.46

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 16/20 0.46
NPC1 O15118 1/20 0.36
MAPT P10636 1/20 0.36
RAB9A P51151 1/20 0.36
MCHR1 Q99705 1/20 0.35
EPHX2 P34913 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3836423 0.82 GRM5 (0.58) GRM5NPC1RAB9A
SCHEMBL3836422 0.82 GRM5 (0.58) GRM5NPC1RAB9A
SCHEMBL3837282 0.82 GRM5 (0.58) GRM5NPC1RAB9A
SCHEMBL3835764 0.80 GRM5 (0.46) GRM5NPC1RAB9AEPHX2
SCHEMBL3860245 0.79 GRM5 (0.52) GRM5
SCHEMBL3836458 0.79 GRM5 (0.52) GRM5
SCHEMBL3836455 0.79 GRM5 (0.52) GRM5
SCHEMBL3841794 0.79 GRM5 (0.46) GRM5RAB9AEPHX2
SCHEMBL3841449 0.79 GRM5 (0.46) GRM5RAB9AEPHX2
SCHEMBL3840495 0.79 GRM5 (0.43) GRM5NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1877367-B1 ACETYLENE DERIVATIVES NOVARTIS AG (CH) 2009-10-14 EP claimed