SCHEMBL3840495

SCHEMBL3840495

O=C(N[C@H]1CC[C@@](O)(C#Cc2cccc(Cl)c2)CC1)Oc1cc2ccccc2o1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 7/20 0.43
RAB9A P51151 3/20 0.37
FAAH O00519 2/20 0.35
NPC1 O15118 3/20 0.35
MAOB P27338 2/20 0.35
EPHX1 P07099 1/20 0.35
PTPRC P08575 1/20 0.35
PTPN2 P17706 1/20 0.35
PTPN1 P18031 1/20 0.35
PTPRB P23467 1/20 0.35
PTPRG P23470 1/20 0.35
ACP1 P24666 1/20 0.35
PTPN3 P26045 1/20 0.35
PTPRM P28827 1/20 0.35
PTPN6 P29350 1/20 0.35
PTPN7 P35236 1/20 0.35
PTPN9 P43378 1/20 0.35
DUSP3 P51452 1/20 0.35
PTPN12 Q05209 1/20 0.35
PTPN11 Q06124 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3376495 0.90 GRM5 (0.43) GRM5RAB9AFAAHNPC1MAOB
SCHEMBL3835764 0.83 GRM5 (0.46) GRM5RAB9ANPC1PTPRCPTPN2
SCHEMBL3836423 0.80 GRM5 (0.58) GRM5RAB9ANPC1
SCHEMBL3837282 0.80 GRM5 (0.58) GRM5RAB9ANPC1
SCHEMBL3836422 0.80 GRM5 (0.58) GRM5RAB9ANPC1
SCHEMBL3841449 0.79 GRM5 (0.46) GRM5RAB9AFAAHPTPRCPTPN2
SCHEMBL3836682 0.79 GRM5 (0.46) GRM5RAB9ANPC1
SCHEMBL3841794 0.79 GRM5 (0.46) GRM5RAB9AFAAHPTPRCPTPN2
SCHEMBL3836458 0.77 GRM5 (0.52) GRM5MAOB
SCHEMBL3860245 0.77 GRM5 (0.52) GRM5MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1877367-B1 ACETYLENE DERIVATIVES NOVARTIS AG (CH) 2009-10-14 EP claimed