SCHEMBL3836901

SCHEMBL3836901

O=C1NCc2cc(F)cc(I)c21

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 3/20 0.37
AURKA O14965 3/20 0.33
CLK4 Q9HAZ1 2/20 0.33
NTRK1 P04629 2/20 0.33
FLT3 P36888 2/20 0.33
GSK3B P49841 2/20 0.33
CA12 O43570 1/20 0.33
CA9 Q16790 1/20 0.33
MKNK2 Q9HBH9 1/20 0.33
DAPK3 O43293 1/20 0.33
PIM1 P11309 1/20 0.33
ROCK1 Q13464 1/20 0.33
KDR P35968 3/20 0.33
PIK3CD O00329 1/20 0.32
PIK3CA P42336 1/20 0.32
PIK3CB P42338 1/20 0.32
TDP2 O95551 1/20 0.32
PARP1 P09874 1/20 0.32
PARP10 Q53GL7 1/20 0.32
MET P08581 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31158957 1.00 GRM5 (0.37) GRM5AURKACLK4NTRK1FLT3
SCHEMBL23089173 0.81 GRM5 (0.37) GRM5AURKACLK4NTRK1FLT3
SCHEMBL23364331 0.81 MKNK2 (0.43) GRM5AURKACLK4NTRK1FLT3
SCHEMBL3840001 0.79 PARP10 (0.36) AURKACLK4NTRK1FLT3GSK3B
SCHEMBL3835512 0.79 KDR (0.41) AURKACLK4NTRK1FLT3GSK3B
SCHEMBL3837295 0.78 AURKA (0.37) AURKACLK4NTRK1FLT3GSK3B
SCHEMBL3835742 0.78 AURKA (0.37) AURKACLK4NTRK1FLT3GSK3B
SCHEMBL31392277 0.78 GRM5 (0.37) GRM5AURKACLK4NTRK1FLT3
SCHEMBL31159152 0.75 GRM5 (0.36) GRM5AURKACLK4NTRK1FLT3
SCHEMBL3840782 0.75 AURKA (0.32) AURKACA12CA9KDRTDP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2108642-A1 JAK INHIBITOR Kyowa Hakko Kirin Co., Ltd. (JP) 2009-10-14 EP disclosed