SCHEMBL3837154

SCHEMBL3837154

O=C(O)N1CCN(c2ccc(Nc3ncc4cnn(C5CCCCCC5)c4n3)cc2)CC1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 13/20 0.56
CCND1 P24385 10/20 0.56
CCND2 P30279 8/20 0.56
CCND3 P30281 8/20 0.56
CDK1 P06493 10/20 0.56
CCNB1 P14635 8/20 0.56
CCNA2 P20248 6/20 0.56
CDK2 P24941 6/20 0.56
CCNE2 O96020 5/20 0.56
CCNE1 P24864 5/20 0.56
CCNA1 P78396 5/20 0.56
CCNB2 O95067 3/20 0.56
CCNB3 Q8WWL7 3/20 0.56
AURKA O14965 9/20 0.55
INSR P06213 1/20 0.55
PDGFRB P09619 1/20 0.55
SRC P12931 1/20 0.55
PDGFRA P16234 1/20 0.55
FLT1 P17948 1/20 0.55
FLT4 P35916 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12639318 0.91 CDK4 (0.67) CDK4CCND1CCND2CCND3CDK1
SCHEMBL12672279 0.91 CDK4 (0.53) CDK4CCND1CCND2CCND3CDK1
SCHEMBL12639370 0.88 CDK1 (0.56) CDK4CCND1CCND2CCND3CDK1
SCHEMBL12639365 0.88 CDK4 (0.54) CDK4CCND1CCND2CCND3CDK1
SCHEMBL1355312 0.88 CDK4 (0.67) CDK4CCND1CCND2CCND3CDK1
SCHEMBL1355734 0.86 CDK4 (0.69) CDK4CCND1CCND2CCND3CDK1
SCHEMBL12639344 0.86 CDK4 (0.69) CDK4CCND1CCND2CCND3CDK1
SCHEMBL12639329 0.86 CDK4 (0.61) CDK4CCND1CCND2CCND3CDK1
SCHEMBL1355087 0.86 CDK4 (0.73) CDK4CCND1CCND2CCND3CDK1
SCHEMBL344014 0.86 CDK4 (0.73) CDK4CCND1CCND2CCND3CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2108020-A2 1-H-PYRAZOLO[3,4B]PYRIMIDINE DERIVATIVES AND THEIR USE AS MODULATORS OF MITOTIC KINASES Biogen Idec MA, Inc. (US) 2009-10-14 EP claimed
WO-2008094602-A2 1-H-PYRAZOLO (3,4B) PYRIMIDINE DERIVATIVES AND THEIR USE AS MODULATORS OF MITOTIC KINASES BIOGEN IDEC MA INC. (US) 2008-08-07 WO claimed