SCHEMBL3837162

SCHEMBL3837162

O=C(CCC1CCCC1)Nc1c(Cl)ccc2nc(N3CCC(OC(=O)O)CC3)ccc12

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 11/20 0.49
KCNQ3 O43525 2/20 0.48
KCNQ2 O43526 2/20 0.48
GBA1 P04062 1/20 0.47
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
ALDH1A1 P00352 1/20 0.38
TP53 P04637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1813063 0.88 P2RX7 (0.51) P2RX7KCNQ3KCNQ2GBA1NPC1
SCHEMBL1804173 0.87 P2RX7 (0.51) P2RX7KCNQ3KCNQ2GBA1NPC1
SCHEMBL1804350 0.85 P2RX7 (0.65) P2RX7KCNQ3KCNQ2GBA1NPC1
SCHEMBL5747310 0.84 P2RX7 (0.54) P2RX7KCNQ3KCNQ2GBA1
SCHEMBL1804596 0.84 P2RX7 (0.54) P2RX7KCNQ3KCNQ2GBA1
SCHEMBL3840972 0.84 P2RX7 (0.54) P2RX7KCNQ3KCNQ2GBA1ALDH1A1
SCHEMBL1801969 0.84 P2RX7 (0.54) P2RX7KCNQ3KCNQ2GBA1ALDH1A1
SCHEMBL3839569 0.81 P2RX7 (0.47) P2RX7
SCHEMBL1802502 0.81 P2RX7 (0.57) P2RX7KCNQ3KCNQ2GBA1
SCHEMBL3839589 0.80 P2RX7 (0.55) P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1633717-B1 P2X7 RECEPTOR ANTAGONISTS AND THEIR USE ASTRAZENECA AB (SE) 2009-10-28 EP claimed