SCHEMBL3837659

SCHEMBL3837659

NS(=O)(=O)c1ccc(NC(=O)Cc2ccc(-c3ccc(Cl)c(Oc4cc(Cl)ccc4Br)c3)cc2)cc1

nearest known ligand 0.60

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CA1 P00915 9/20 0.60
CA2 P00918 9/20 0.60
CA12 O43570 8/20 0.60
CA9 Q16790 8/20 0.60
RORC P51449 4/20 0.53
POLB P06746 2/20 0.51
CA5A P35218 2/20 0.48
CA7 P43166 2/20 0.48
CA5B Q9Y2D0 2/20 0.48
CA14 Q9ULX7 1/20 0.48
P2RX4 Q99571 2/20 0.47
LMNA P02545 2/20 0.46
ALDH1A1 P00352 1/20 0.46
HTT P42858 1/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2638624 0.92 CA1 (0.61) CA1CA2CA12CA9RORC
SCHEMBL4603317 0.87 CA1 (0.61) CA1CA2CA12CA9RORC
SCHEMBL3837658 0.86 CA12 (0.53) CA1CA2CA12CA9RORC
SCHEMBL2639161 0.83 CA2 (0.59) CA1CA2CA12CA9RORC
SCHEMBL2639656 0.82 CA1 (0.58) CA1CA2CA12CA9RORC
SCHEMBL2640024 0.81 CA1 (0.59) CA1CA2CA12CA9RORC
SCHEMBL2639462 0.81 CA1 (0.56) CA1CA2CA12CA9RORC
SCHEMBL14625926 0.80 P2RX4 (0.59) CA1CA2CA12CA9POLB
SCHEMBL2638691 0.75 CA1 (0.61) CA1CA2CA12CA9RORC
SCHEMBL13581454 0.74 CA1 (0.70) CA1CA2CA12CA9RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1742908-B1 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS HOFFMANN LA ROCHE (CH) 2009-11-11 EP disclosed