SCHEMBL3838017

SCHEMBL3838017

COC(=O)CCCNC(=O)Nc1nc(C)c(-c2ccnc(N3CCOCC3)c2)s1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.45
ALDH1A1 P00352 1/20 0.45
TSHR P16473 1/20 0.45
CLK1 P49759 1/20 0.45
RAB9A P51151 1/20 0.45
PIK3CA P42336 8/20 0.42
PIK3CG P48736 7/20 0.42
PIK3CD O00329 7/20 0.42
PIK3CB P42338 5/20 0.42
RAF1 P04049 6/20 0.41
BRAF P15056 6/20 0.41
PI4KB Q9UBF8 2/20 0.41
DYRK3 O43781 1/20 0.41
MAP4K4 O95819 1/20 0.41
CLK2 P49760 1/20 0.41
DYRK1A Q13627 1/20 0.41
MINK1 Q8N4C8 1/20 0.41
CLK4 Q9HAZ1 1/20 0.41
ADORA2A P29274 1/20 0.40
ADORA1 P30542 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1884162 0.94 PIK3CA (0.46) NPC1ALDH1A1TSHRCLK1RAB9A
SCHEMBL1891436 0.89 PIK3CA (0.47) NPC1ALDH1A1TSHRCLK1RAB9A
SCHEMBL1888686 0.81 PIK3CG (0.60) NPC1ALDH1A1TSHRCLK1RAB9A
SCHEMBL5048755 0.75 NPC1 (0.51) NPC1ALDH1A1TSHRCLK1RAB9A
SCHEMBL12991910 0.72 PIK3CG (0.50) NPC1ALDH1A1RAB9APIK3CAPIK3CG
SCHEMBL1889933 0.71 CDK2 (0.43) ADORA2AADORA1
SCHEMBL12991926 0.70 NPC1 (0.53) NPC1ALDH1A1TSHRCLK1RAB9A
SCHEMBL8236670 0.70 PIK3CA (0.54) NPC1CLK1RAB9APIK3CAPIK3CD
SCHEMBL1885306 0.70 KARS1 (0.48) RAF1BRAFADORA2AADORA1
SCHEMBL28407628 0.69 ADORA2A (0.62) ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1622897-B1 INHIBITORS OF PHOSPHATIDYLINOSITOL 3-KINASE NOVARTIS AG (CH) 2009-10-14 EP disclosed