SCHEMBL3840665

SCHEMBL3840665

CCCOc1cc2c(c(-c3cc4ccccc4[nH]3)c1)C(=O)NC2

nearest known ligand 0.60

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDR P35968 16/20 0.60
AURKA O14965 11/20 0.60
CDK1 P06493 1/20 0.45
CHEK1 O14757 1/20 0.40
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38
RAB9A P51151 1/20 0.38
KMT2A Q03164 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
CTSV O60911 1/20 0.37
CTSL P07711 1/20 0.37
HRH3 Q9Y5N1 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3840660 0.83 KDR (0.62) KDRAURKACDK1CHEK1KDM4E
SCHEMBL3836059 0.82 AURKA (0.54) KDRAURKA
Hydrochloric Acid SCHEMBL3837263 0.77 KDR (0.54) KDRAURKACDK1CHEK1MEN1
SCHEMBL3835222 0.76 KDR (0.62) KDRAURKACDK1CHEK1KDM4E
SCHEMBL14468698 0.76 KDR (0.83) KDRAURKACDK1CTSVCTSL
SCHEMBL5333071 0.75 KDR (1.00) KDRAURKACDK1CHEK1KDM4E
SCHEMBL5329803 0.74 KDR (0.77) KDRAURKACDK1KDM4EMEN1
SCHEMBL3835801 0.71 ELANE (0.37) KDRAURKAALDH1A1MAPT
Hydrochloric Acid SCHEMBL3839444 0.70 KDR (0.60) KDRAURKACDK1CHEK1KDM4E
SCHEMBL5327042 0.69 KDR (1.00) KDRAURKACDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2108642-A1 JAK INHIBITOR Kyowa Hakko Kirin Co., Ltd. (JP) 2009-10-14 EP disclosed