SCHEMBL3842664

SCHEMBL3842664

O=[C]NCc1ccc(C(F)(F)F)nc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.48
MAOA P21397 1/20 0.48
MAOB P27338 1/20 0.48
TRPV1 Q8NER1 1/20 0.45
TRPV4 Q9HBA0 1/20 0.44
DAO P14920 3/20 0.43
NAMPT P43490 2/20 0.42
KCNQ3 O43525 1/20 0.41
KCNQ2 O43526 1/20 0.41
KCNQ4 P56696 1/20 0.41
KCNQ5 Q9NR82 1/20 0.41
CNR1 P21554 2/20 0.39
CSF1R P07333 2/20 0.39
CNR2 P34972 1/20 0.39
CYP2C19 P33261 1/20 0.39
LCK P06239 1/20 0.39
PGR P06401 1/20 0.39
CHRM2 P08172 1/20 0.39
HTR1A P08908 1/20 0.39
ADRA2A P08913 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6245504 0.79 KDM1A (0.50) KDM1AMAOAMAOBTRPV1TRPV4
SCHEMBL297140 0.79 KDM1A (0.50) KDM1AMAOAMAOBTRPV1TRPV4
SCHEMBL29196353 0.78 KDM1A (0.47) KDM1AMAOAMAOBTRPV1TRPV4
SCHEMBL30887515 0.78 KDM1A (0.47) KDM1AMAOAMAOBTRPV1TRPV4
SCHEMBL3842669 0.78 KDM1A (0.47) KDM1AMAOAMAOBTRPV1TRPV4
SCHEMBL14614919 0.77 KDM1A (0.49) KDM1AMAOAMAOBTRPV1TRPV4
Hydrochloric Acid SCHEMBL20581296 0.77 KDM1A (0.49) KDM1AMAOAMAOBTRPV1TRPV4
SCHEMBL22501639 0.77 TRPV1 (0.52) KDM1AMAOAMAOBTRPV1DAO
SCHEMBL13061262 0.76 KDM1A (0.48) KDM1AMAOAMAOBTRPV1TRPV4
SCHEMBL452178 0.76 TRPV4 (0.52) KDM1AMAOAMAOBTRPV1TRPV4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1979354-B1 DIAZA-SPIRO-[4, 5]-DECANES USEFUL AS PESTICIDES SYNGENTA PARTICIPATIONS AG (CH) 2009-11-11 EP disclosed
EP-2089034-A1 NOVEL USES Intra-Cellular Therapies, Inc. (US) 2009-08-19 EP disclosed
EP-2081431-A1 ORGANIC COMPOUNDS Intra-Cellular Therapies, Inc. (US) 2009-07-29 EP disclosed
WO-2008070095-A1 NOVEL USES INTRA-CELLULAR THERAPIES, INC. (US) 2008-06-12 WO disclosed
WO-2008063505-A1 ORGANIC COMPOUNDS INTRA-CELLULAR THERAPIES, INC. (US) 2008-05-29 WO disclosed