SCHEMBL3843083

SCHEMBL3843083

O=C(O)N1CCc2cc(OS(=O)(=O)C(F)(F)F)ccc2C1

nearest known ligand 0.57

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 7/20 0.57
ESR1 P03372 6/20 0.57
ABHD6 Q9BV23 3/20 0.52
DRD2 P14416 8/20 0.46
DRD3 P35462 8/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA7 P43166 1/20 0.46
CA9 Q16790 1/20 0.46
CA14 Q9ULX7 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7974143 0.95 ESR1 (0.51) ESR2ESR1ABHD6DRD2DRD3
SCHEMBL30548173 0.85 ESR2 (0.65) ESR2ESR1ABHD6DRD2DRD3
SCHEMBL587484 0.85 ESR2 (0.65) ESR2ESR1ABHD6DRD2DRD3
SCHEMBL3781320 0.84 HRH3 (0.52) ESR2ESR1ABHD6DRD2DRD3
SCHEMBL6160274 0.81 TMEM97 (0.60) ESR2ESR1ABHD6DRD3
SCHEMBL29052398 0.81 ESR1 (0.41) ESR2ESR1ABHD6DRD2DRD3
SCHEMBL13094748 0.81 DRD1 (0.56) ESR2ESR1DRD2DRD3
SCHEMBL7798191 0.81 ITGB3 (0.54) ESR2ESR1DRD2DRD3
SCHEMBL1650187 0.80 NR1H2 (0.63) ESR2ESR1ABHD6DRD2DRD3
SCHEMBL11295872 0.80 ESR1 (0.71) ESR2ESR1ABHD6DRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116507326-A Compounds as GLP-1R agonists 拓臻制药公司 2023-07-28 CN disclosed
EP-3053917-A1 T-TYPE CALCIUM CHANNEL BLOCKER Nissan Chemical Industries, Ltd. (JP) 2016-08-10 EP disclosed
EP-1998620-A4 PIPERAZINYL OXOALKYL TETRAHYDROISOQUINOLINES AND RELATED ANALOGUES NEUROGEN CORP (US) 2009-09-02 EP disclosed
EP-1998620-A2 PIPERAZINYL OXOALKYL TETRAHYDROISOQUINOLINES AND RELATED ANALOGUES Neurogen Corporation (US) 2008-12-10 EP disclosed
WO-2007106349-A2 PIPERAZINYL OXOALKYL TETRAHYDROISOQUINOLINES AND RELATED ANALOGUES NEUROGEN CORPORATION (US) 2007-09-20 WO disclosed
US-5700809-A Pyrrolo-pyridine derivatives MERCK SHARP & DOHME, LTD. (GB) 1997-12-23 US disclosed