SCHEMBL3845293

SCHEMBL3845293

Clc1cc(-c2cnn(C(c3ccccc3)(c3ccccc3)c3ccccc3)c2)cn2c(-c3nccs3)cnc12

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KDR P35968 1/20 0.42
MET P08581 1/20 0.35
SLC16A3 O15427 1/20 0.33
SLC16A1 P53985 1/20 0.33
MCTS1 Q9ULC4 1/20 0.33
PDPK1 O15530 1/20 0.33
KCNN4 O15554 1/20 0.30
KCNA3 P22001 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3847544 0.83 MET (0.37) KDRMETKCNN4KCNA3
SCHEMBL3845295 0.82 KDR (0.35) KDRMET
SCHEMBL3844953 0.79 MET (0.36) METKCNN4KCNA3
SCHEMBL3847999 0.73 KCNN4 (0.38) METKCNN4KCNA3
Hydrochloric Acid SCHEMBL3848522 0.72 CHEK1 (0.40) KDR
SCHEMBL3847947 0.70 KDR (0.38) KDRMET
SCHEMBL3847154 0.69 KDR (0.37) KDR
SCHEMBL3848204 0.68 KDR (0.41) KDRPDPK1
SCHEMBL3847823 0.67 KDR (0.35) KDR
Hydrochloric Acid SCHEMBL3855523 0.67 KDR (0.36) KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2048142-A2 Nitrogen-containing condensed cyclic compound having a pyrazolyl group as a substituent group and pharmaceutical composition thereof Eisai R&D Management Co., Ltd. (JP) 2009-04-15 EP disclosed
EP-1382603-B1 NITROGENOUS FUSED-RING COMPOUND HAVING PYRAZOLYL GROUP AS SUBSTITUENT AND MEDICINAL COMPOSITION THEREOF EISAI R&D MAN CO LTD (JP) 2008-07-23 EP disclosed
US-7074801-B1 Nitrogen-containing condensed cyclic compound having a pyrazolyl group as a substituent group and pharmaceutical composition thereof EISAI CO., LTD. (JP) 2006-07-11 US disclosed
EP-1382603-A1 NITROGENOUS FUSED−RING COMPOUND HAVING PYRAZOLYL GROUP AS SUBSTITUENT AND MEDICINAL COMPOSITION THEREOF Eisai Co., Ltd. (JP) 2004-01-21 EP disclosed