SCHEMBL3846552

SCHEMBL3846552

CC(=O)c1ccc2ccc(N(C(=O)OC(C)(C)C)C(Br)C=CCl)cc2c1

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.36
CYP17A1 P05093 1/20 0.32
CYP3A4 P08684 1/20 0.32
MEN1 O00255 1/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
KMT2A Q03164 1/20 0.31
ALDH1A1 P00352 1/20 0.30
MAPT P10636 1/20 0.30
HPGD P15428 1/20 0.30
GABRB1 P18505 1/20 0.30
GABRB2 P47870 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3851122 0.87 MEN1 (0.37) MEN1KMT2AALDH1A1GABRB1GABRB2
SCHEMBL3566610 0.83 AKR1C3 (0.33)
SCHEMBL3559266 0.83 NCEH1 (0.35)
SCHEMBL3564219 0.80 NCEH1 (0.36)
SCHEMBL3559616 0.80 AKR1C3 (0.36)
SCHEMBL3827000 0.77 CYP2A6 (0.45) CYP2A6CYP17A1CYP3A4MEN1NPC1
SCHEMBL3557776 0.76 CNR2 (0.46) MEN1KMT2AMAPT
SCHEMBL16682552 0.71 RAB9A (0.43) CYP2A6CYP17A1CYP3A4MEN1NPC1
SCHEMBL7447861 0.65 MEN1 (0.40) MEN1KMT2AALDH1A1GABRB1GABRB2
SCHEMBL16682553 0.65 MAPT (0.39) CYP2A6CYP17A1CYP3A4MEN1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1809603-A4 NITROBENZINDOLES AND THEIR USE IN CANCER THERAPY AUCKLAND UNISERVICES LTD (NZ) 2009-09-02 EP disclosed
EP-1809603-A1 NITROBENZINDOLES AND THEIR USE IN CANCER THERAPY Auckland Uniservices Limited (NZ) 2007-07-25 EP disclosed
WO-2006043839-A1 NITROBENZINDOLES AND THEIR USE IN CANCER THERAPY AUCKLAND UNISERVICES LIMITED (NZ) 2006-04-27 WO disclosed