SCHEMBL3847065

SCHEMBL3847065

CSc1ccc(-c2cnc3ccc(-c4cn(C(c5ccccc5)(c5ccccc5)c5ccccc5)nc4-c4ccc(CN(C)C)cc4)cn23)s1

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
FLT3 P36888 10/20 0.34
AXL P30530 2/20 0.31
NTRK1 P04629 1/20 0.31
NTRK3 Q16288 1/20 0.31
NTRK2 Q16620 1/20 0.31
EED O75530 1/20 0.31
SLC2A1 P11166 1/20 0.30
TYRO3 Q06418 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3846331 0.91 FYN (0.38) FLT3
SCHEMBL3849419 0.90 FLT3 (0.36) FLT3
SCHEMBL3845544 0.88 FLT3 (0.44) FLT3
SCHEMBL3850681 0.88 FLT3 (0.37) FLT3
SCHEMBL3848127 0.86 FLT3 (0.40) FLT3AXLNTRK1NTRK3NTRK2
SCHEMBL3848455 0.86 MKNK1 (0.38) FLT3
SCHEMBL3853072 0.85 FLT3 (0.49) FLT3
SCHEMBL4717164 0.85 FLT3 (0.32) FLT3
SCHEMBL3846538 0.84 FLT3 (0.36) FLT3SLC2A1
SCHEMBL3851974 0.84 TGFBR1 (0.38) FLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2048142-A2 Nitrogen-containing condensed cyclic compound having a pyrazolyl group as a substituent group and pharmaceutical composition thereof Eisai R&D Management Co., Ltd. (JP) 2009-04-15 EP disclosed
EP-1382603-B1 NITROGENOUS FUSED-RING COMPOUND HAVING PYRAZOLYL GROUP AS SUBSTITUENT AND MEDICINAL COMPOSITION THEREOF EISAI R&D MAN CO LTD (JP) 2008-07-23 EP disclosed
US-7074801-B1 Nitrogen-containing condensed cyclic compound having a pyrazolyl group as a substituent group and pharmaceutical composition thereof EISAI CO., LTD. (JP) 2006-07-11 US disclosed
EP-1382603-A1 NITROGENOUS FUSED−RING COMPOUND HAVING PYRAZOLYL GROUP AS SUBSTITUENT AND MEDICINAL COMPOSITION THEREOF Eisai Co., Ltd. (JP) 2004-01-21 EP disclosed