SCHEMBL3847804

SCHEMBL3847804

COc1ccc(C2(C)CCCc3cc(O)ccc3C2)cc1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 4/20 0.42
ESR2 Q92731 4/20 0.41
NPC1 O15118 1/20 0.39
POLB P06746 1/20 0.39
RAB9A P51151 1/20 0.39
KDM1A O60341 1/20 0.39
MIF P14174 1/20 0.38
SIGMAR1 Q99720 1/20 0.37
ADRA2A P08913 1/20 0.37
STS P08842 1/20 0.37
LTA4H P09960 1/20 0.37
CYP26A1 O43174 1/20 0.36
CES2 O00748 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3657421 0.92 KDM1A (0.45) ESR1KDM1AMIFADRA2ACYP26A1
SCHEMBL3649238 0.89 KDM1A (0.49) KDM1ASIGMAR1ADRA2A
SCHEMBL3649486 0.89 ESR1 (0.43) ESR1ESR2
SCHEMBL13875403 0.89 ESR1 (0.43) ESR1ESR2
SCHEMBL3655256 0.81 ESR2 (0.47) ESR1ESR2NPC1POLBRAB9A
SCHEMBL3652676 0.80 ESR1 (0.39) ESR1NPC1POLBRAB9AKDM1A
SCHEMBL3653751 0.79 OPRD1 (0.54) ESR1ESR2
SCHEMBL3844606 0.78 ESR2 (0.39) ESR1ESR2
SCHEMBL3647466 0.77 ESR1 (0.40) ESR1ESR2
SCHEMBL3853852 0.77 ESR1 (0.39) ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090099250-A1 BENZOCYCLOHEPTENE DERIVATIVES AS ESTROGENS HAVING SELECTIVE ACTIVITY BAYER SCHERING PHARMA AG (DE) 2009-04-16 US claimed
US-20090099250-A1 BENZOCYCLOHEPTENE DERIVATIVES AS ESTROGENS HAVING SELECTIVE ACTIVITY BAYER SCHERING PHARMA AG (DE) 2009-04-16 US disclosed
EP-2048126-A1 Benzocycloheptane derivatives as selectively active oestrogens Bayer Schering Pharma AG (DE) 2009-04-15 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090099250-A1 BENZOCYCLOHEPTENE DERIVATIVES AS ESTROGENS HAVING SELECTIVE ACTIVITY CYP19A1, HSD17B11, CYP21A2 ESR1 4/4885ESR2 23/4885NPC1 416/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.