SCHEMBL3848486

SCHEMBL3848486

O=C(Nc1nc2ccc(F)cc2s1)c1ccc(-c2cnc3ccc(-c4cn[nH]c4)cn23)cc1F

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.46
SMN1; SMN2 Q16637 3/20 0.46
KDR P35968 4/20 0.45
NPC1 O15118 4/20 0.42
RAB9A P51151 4/20 0.42
HTT P42858 2/20 0.42
POLB P06746 1/20 0.42
PKM P14618 1/20 0.42
AGTR1 P30556 1/20 0.42
OPRK1 P41145 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
LRRK2 Q5S007 2/20 0.42
KDM4E B2RXH2 2/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
ROCK2 O75116 1/20 0.41
OTUD7B Q6GQQ9 1/20 0.41
HSD17B1 P14061 1/20 0.41
HSD17B2 P37059 1/20 0.41
PTGES O14684 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5852278 0.99 MAPT (0.46) MAPTSMN1; SMN2KDRNPC1RAB9A
Hydrochloric Acid SCHEMBL3846532 0.89 DYRK1A (0.45) NPC1RAB9AOTUD7BHSD17B1HSD17B2
SCHEMBL4712318 0.83 KDM4E (0.41) MAPTPOLBLRRK2KDM4EROCK2
Hydrochloric Acid SCHEMBL3849122 0.83 KDM4E (0.40) MAPTPOLBLRRK2KDM4EROCK2
Hydrochloric Acid SCHEMBL3845647 0.83 LRRK2 (0.45) NPC1RAB9ATDP1LRRK2KDM4E
Hydrochloric Acid SCHEMBL3850519 0.82 GSK3B (0.42) SMN1; SMN2NPC1RAB9AROCK2DYRK1A
SCHEMBL3855822 0.82 FLT3 (0.41) MAPTNPC1RAB9APOLBMEN1
SCHEMBL3851356 0.82 KDR (0.46) MAPTSMN1; SMN2KDRNPC1RAB9A
Hydrochloric Acid SCHEMBL5853314 0.81 FLT3 (0.41) MAPTNPC1RAB9APOLBMEN1
Hydrochloric Acid SCHEMBL3849246 0.81 FLT3 (0.39) SMN1; SMN2NPC1RAB9AROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2048142-A2 Nitrogen-containing condensed cyclic compound having a pyrazolyl group as a substituent group and pharmaceutical composition thereof Eisai R&D Management Co., Ltd. (JP) 2009-04-15 EP disclosed
EP-1382603-B1 NITROGENOUS FUSED-RING COMPOUND HAVING PYRAZOLYL GROUP AS SUBSTITUENT AND MEDICINAL COMPOSITION THEREOF EISAI R&D MAN CO LTD (JP) 2008-07-23 EP disclosed