SCHEMBL3855822

SCHEMBL3855822

O=C(Nc1nccs1)c1ccc(-c2cnc3ccc(-c4cn[nH]c4)cn23)cc1F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FLT3 P36888 2/20 0.41
ROCK2 O75116 1/20 0.40
ROCK1 Q13464 1/20 0.40
NRAS P01111 1/20 0.40
NPC1 O15118 4/20 0.38
RAB9A P51151 4/20 0.38
KCNMA1 Q12791 1/20 0.38
CHEK1 O14757 5/20 0.38
CHEK2 O96017 1/20 0.38
ABL1 P00519 1/20 0.38
MET P08581 1/20 0.37
PTK6 Q13882 1/20 0.37
AURKB Q96GD4 1/20 0.37
MAPT P10636 2/20 0.37
POLB P06746 1/20 0.37
LMNA P02545 1/20 0.37
HPGD P15428 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
MAPK1 P28482 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5853314 0.99 FLT3 (0.41) FLT3ROCK2ROCK1NRASNPC1
Hydrochloric Acid SCHEMBL3849246 0.87 FLT3 (0.39) FLT3ROCK2ROCK1NRASNPC1
Hydrochloric Acid SCHEMBL3846959 0.85 ALDH1A1 (0.45) FLT3ROCK2ROCK1NRASPTK6
Hydrochloric Acid SCHEMBL3850519 0.85 GSK3B (0.42) FLT3ROCK2ROCK1NRASNPC1
Hydrochloric Acid SCHEMBL3854256 0.84 ALDH1A1 (0.46) FLT3NRASNPC1RAB9AMAPT
Hydrochloric Acid SCHEMBL3845647 0.83 LRRK2 (0.45) FLT3ROCK2ROCK1NRASNPC1
Hydrochloric Acid SCHEMBL3845019 0.83 FLT3 (0.43) FLT3ROCK2NRASPTK6AURKB
SCHEMBL4712318 0.82 KDM4E (0.41) FLT3ROCK2ROCK1NRASCHEK1
SCHEMBL3848486 0.82 MAPT (0.46) ROCK2NPC1RAB9AMAPTPOLB
SCHEMBL4715804 0.82 LOXL2 (0.43) FLT3ROCK2ROCK1NRASNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2048142-A2 Nitrogen-containing condensed cyclic compound having a pyrazolyl group as a substituent group and pharmaceutical composition thereof Eisai R&D Management Co., Ltd. (JP) 2009-04-15 EP disclosed
EP-1382603-B1 NITROGENOUS FUSED-RING COMPOUND HAVING PYRAZOLYL GROUP AS SUBSTITUENT AND MEDICINAL COMPOSITION THEREOF EISAI R&D MAN CO LTD (JP) 2008-07-23 EP disclosed