SCHEMBL3854285

SCHEMBL3854285

[CH2]c1ccccc1P(=O)(O)O

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.44
CA4 P22748 1/20 0.44
CA5A P35218 1/20 0.44
PTK2B Q14289 5/20 0.44
POLB P06746 3/20 0.44
NPC1 O15118 2/20 0.44
ALDH1A1 P00352 1/20 0.42
RAB9A P51151 1/20 0.42
ALPG P10696 1/20 0.41
KDM4E B2RXH2 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
ALOX15 P16050 1/20 0.37
TSHR P16473 1/20 0.37
MAPT P10636 1/20 0.36
SRC P12931 2/20 0.34
CFTR P13569 1/20 0.34
FDPS P14324 1/20 0.34
PTPN1 P18031 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2173729 0.81 CA2 (0.55) CA2CA4CA5APTK2BPOLB
SCHEMBL29733396 0.81 CA2 (0.55) CA2CA4CA5APTK2BPOLB
SCHEMBL4956835 0.74 CA2 (0.48) CA2CA4CA5APTK2BPOLB
SCHEMBL1227487 0.72 CYP3A4 (0.52) CA2CA4CA5APTK2BPOLB
SCHEMBL846360 0.70 CA2 (0.44) CA2CA4CA5APTK2BPOLB
SCHEMBL3889145 0.70 CA2 (0.44) CA2CA4CA5APTK2BPOLB
SCHEMBL7812902 0.70 CA2 (0.44) CA2CA4CA5APTK2BPOLB
SCHEMBL232481 0.70 CA2 (0.44) CA2CA4CA5APTK2BPOLB
SCHEMBL11350253 0.70 CYP3A4 (0.50) CA2CA4CA5APTK2BPOLB
SCHEMBL3365510 0.70 CA2 (0.44) CA2CA4CA5APTK2BPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114716386-A Novel exosome inhibitor and preparation method thereof 北京和理咨询有限公司 2022-07-08 CN claimed
WO-2008031888-A2 CONDENSED PYRIMIDINONES ACTIVE ON GLUTAMATERGIC RECEPTORS CAMPIANI GIUSEPPE (IT) 2008-03-20 WO claimed
CN-116622005-A Polymer prodrug compound and preparation method thereof, and polymer prodrug micelle and preparation method thereof 成都普康生物科技有限公司 2023-08-22 CN disclosed
CN-114716386-A Novel exosome inhibitor and preparation method thereof 北京和理咨询有限公司 2022-07-08 CN disclosed
CN-107847607-B Aptamer conjugate of paclitaxel or derivative thereof, and preparation method and application thereof 北京盈科瑞创新医药股份有限公司 2020-11-20 CN disclosed
CN-110483531-B Water-soluble porphyrin alkene derivative, preparation method, antitumor drug and application 李德芳 2020-08-04 CN disclosed
CN-108627647-A A kind of detection of posttranslational modification proteomics and quantitative approach 四川大学 2018-10-09 CN disclosed
EP-1730228-B1 NANO-COMPOSITE AND METHOD THEREOF BRIDGESTONE CORP (JP) 2012-08-15 EP disclosed
US-7579398-B2 Nano-composite and compositions therefrom BRIDGESTONE CORPORATION (JP) 2009-08-25 US disclosed
US-7572855-B2 Nano-composite and compositions manufactured thereof BRIDGESTONE CORPORATION (JP) 2009-08-11 US disclosed
US-20090182087-A1 NANO-COMPOSITE AND COMPOSITIONS THEREFROM BRIDGESTONE CORPORATION (JP) 2009-07-16 US disclosed
WO-2008031888-A2 CONDENSED PYRIMIDINONES ACTIVE ON GLUTAMATERGIC RECEPTORS CAMPIANI GIUSEPPE (IT) 2008-03-20 WO disclosed
EP-1730228-A1 NANO-COMPOSITE AND METHOD THEREOF Bridgestone Corporation (JP) 2006-12-13 EP disclosed
US-20060173115-A1 Nano-composite and compositions manufactured thereof BRIDGESTONE CORPORATION (JP) 2006-08-03 US disclosed
WO-2005095506-A1 NANO-COMPOSITE AND METHOD THEREOF BRIDGESTONE CORPORATION (JP) 2005-10-13 WO disclosed
US-20020055536-A1 System and method for structure-based drug design that includes accurate prediction of binding free energy DEWITTE ROBERT S (US) 2002-05-09 US disclosed
EP-1140737-A2 SYSTEM AND METHOD FOR STRUCTURE-BASED DRUG DESIGN THAT INCLUDES ACCURATE PREDICTION OF BINDING FREE ENERGY HARVARD UNIVERSITY (US) 2001-10-10 EP disclosed
WO-2000039751-A2 SYSTEM AND METHOD FOR STRUCTURE-BASED DRUG DESIGN THAT INCLUDES ACCURATE PREDICTION OF BINDING FREE ENERGY HARVARD UNIVERSITY (US) 2000-07-06 WO disclosed
US-5449736-A Heat resistant and hydrophobic fluids as dielectrics RESEARCH FOUNDATION OF THE STATE OF NEW YORK (US) 1995-09-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020055536-A1 System and method for structure-based drug design that includes accurate prediction of binding free energy ABCG2, LSS, FARS2 CA2 4261/4885CA4 4112/4885CA5A 2632/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.