SCHEMBL3855867

SCHEMBL3855867

[CH2]c1ccc(-c2nn(C(c3ccccc3)(c3ccccc3)c3ccccc3)cc2-c2ccc3ncc(-c4ccccn4)n3c2)cc1

nearest known ligand 0.40

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 19/20 0.40
TGFBR2 P37173 1/20 0.39
IRAK4 Q9NWZ3 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3846170 0.91 TGFBR1 (0.46) TGFBR1TGFBR2IRAK4
SCHEMBL3846843 0.90 TGFBR1 (0.41) TGFBR1TGFBR2
SCHEMBL3852272 0.90 TGFBR1 (0.41) TGFBR1TGFBR2
SCHEMBL3847481 0.90 TGFBR1 (0.40) TGFBR1TGFBR2
SCHEMBL3846055 0.90 TGFBR1 (0.42) TGFBR1TGFBR2
SCHEMBL3846122 0.88 FYN (0.42) TGFBR1TGFBR2
SCHEMBL3854925 0.88 TGFBR1 (0.39) TGFBR1TGFBR2
SCHEMBL3847225 0.88 TGFBR1 (0.43) TGFBR1TGFBR2
SCHEMBL4712454 0.88 TGFBR1 (0.39) TGFBR1TGFBR2
SCHEMBL3849616 0.88 TGFBR1 (0.39) TGFBR1TGFBR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2048142-A2 Nitrogen-containing condensed cyclic compound having a pyrazolyl group as a substituent group and pharmaceutical composition thereof Eisai R&D Management Co., Ltd. (JP) 2009-04-15 EP disclosed