SCHEMBL3857538

SCHEMBL3857538

Fc1cc(Cl)cc(Br)c1.Fc1cc(Cl)ccc1Br

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.35
RAB9A P51151 3/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
HPGD P15428 1/20 0.35
EPAS1 Q99814 9/20 0.33
KDM1A O60341 2/20 0.33
KCNH2 Q12809 2/20 0.33
KDM1B Q8NB78 1/20 0.33
GRM2 Q14416 1/20 0.31
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30
GAA P10253 1/20 0.30
KMT2A Q03164 1/20 0.30
ACLY P53396 1/20 0.30
MDM2 Q00987 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29387311 0.84
SCHEMBL118511 0.84
SCHEMBL264105 0.82
SCHEMBL29602146 0.82
SCHEMBL20293122 0.80 TSHR (0.35) EPAS1
Boric Acid SCHEMBL2464038 0.74 EPAS1 (0.32) EPAS1
SCHEMBL17514808 0.68 KMO (0.39) NPC1RAB9ASMN1; SMN2GRM2
SCHEMBL29358544 0.68
SCHEMBL692283 0.68
SCHEMBL14413 0.67

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1742908-B1 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS HOFFMANN LA ROCHE (CH) 2009-11-11 EP disclosed