SCHEMBL3862995

SCHEMBL3862995

C[Si](C)(C)c1cc(-c2ccc(Br)cc2)n(-c2ccc(S(N)(=O)=O)cc2)n1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 15/20 0.67
PTGS1 P23219 5/20 0.67
CA1 P00915 4/20 0.65
CA2 P00918 4/20 0.65
CA9 Q16790 3/20 0.65
MMP2 P08253 1/20 0.55
CYP2C9 P11712 3/20 0.54
PDPK1 O15530 2/20 0.54
PTGES O14684 1/20 0.54
HDAC3 O15379 1/20 0.54
CA12 O43570 1/20 0.54
PDE5A O76074 1/20 0.54
ABCB11 O95342 1/20 0.54
MT-CO2 P00403 1/20 0.54
LMNA P02545 1/20 0.54
CA3 P07451 1/20 0.54
CYP3A4 P08684 1/20 0.54
ALOX5 P09917 1/20 0.54
ADORA3 P0DMS8 1/20 0.54
CYP2D6 P10635 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3869967 0.89 PTGS2 (0.68) PTGS2PTGS1CA1CA2CA9
SCHEMBL8121677 0.83 PTGS2 (0.88) PTGS2PTGS1CA1CA2CA9
SCHEMBL3900112 0.80 PTGS2 (1.00) PTGS2PTGS1CA1CA2CA9
SCHEMBL13752026 0.80 PTGS2 (0.64) PTGS2PTGS1CA1CA2CA9
SCHEMBL27485627 0.79 PTGS2 (0.69) PTGS2PTGS1CA1CA2CA9
SCHEMBL6531306 0.79 CA9 (1.00) PTGS2PTGS1CA1CA2CA9
SCHEMBL6350781 0.79 PTGS2 (0.69) PTGS2PTGS1CA1CA2CA9
SCHEMBL6341745 0.79 PTGS2 (0.78) PTGS2PTGS1CA1CA2CA9
SCHEMBL6531664 0.79 PTGS2 (0.78) PTGS2PTGS1CA1CA2CA9
SCHEMBL8119659 0.78 PTGS2 (0.79) PTGS2PTGS1CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7521435-B2 Silicon containing compounds having selective COX-2 inhibitory activity and methods of making and using the same PHARMA DIAGNOSTICS, N.V. (BE) 2009-04-21 US claimed