Ensulizole

Ensulizole

SCHEMBL38724

O=S(=O)(O)c1ccc2nc(-c3ccccc3)[nH]c2c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 1/20 1.00
NPBWR1 P48145 2/20 0.74
SCD O00767 4/20 0.71
CYP2C9 P11712 3/20 0.66
CYP2C19 P33261 3/20 0.66
CYP1A2 P05177 2/20 0.66
CYP3A4 P08684 3/20 0.63
CYP2D6 P10635 1/20 0.63
MAPT P10636 7/20 0.60
TP53 P04637 4/20 0.60
CHEK2 O96017 2/20 0.60
MEN1 O00255 2/20 0.58
KMT2A Q03164 2/20 0.58
SMN1; SMN2 Q16637 3/20 0.58
NPC1 O15118 2/20 0.58
RAB9A P51151 2/20 0.58
KDM4E B2RXH2 2/20 0.57
ALDH1A1 P00352 2/20 0.57
HPGD P15428 2/20 0.57
GLA P06280 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ensulizole SCHEMBL7751558 1.00 HDAC6 (1.00) HDAC6NPBWR1SCDCYP2C9CYP2C19
Ensulizole SCHEMBL1276071 0.99 HDAC6 (0.97) HDAC6NPBWR1SCDCYP2C9CYP2C19
Ensulizole SCHEMBL28708898 0.99 HDAC6 (0.97) HDAC6NPBWR1SCDCYP2C9CYP2C19
Ensulizole SCHEMBL17351654 0.99 HDAC6 (0.97) HDAC6NPBWR1SCDCYP2C9CYP2C19
SCHEMBL30884657 0.97 HDAC6 (0.94) HDAC6NPBWR1SCDCYP2C9CYP2C19
Ensulizole SCHEMBL27885504 0.97 HDAC6 (0.94) HDAC6NPBWR1SCDCYP2C9CYP2C19
Ensulizole SCHEMBL30504101 0.95 HDAC6 (0.90) HDAC6NPBWR1SCDCYP2C9CYP2C19
Ensulizole SCHEMBL1072605 0.93 HDAC6 (0.87) HDAC6NPBWR1SCDCYP2C9CYP2C19
SCHEMBL490323 0.92 HDAC6 (0.86) HDAC6NPBWR1SCDCYP2C9CYP2C19
SCHEMBL5178280 0.92 HDAC6 (0.84) HDAC6NPBWR1SCDCYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 12584 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-122070479-A Ultrasonic indicating device and method for monitoring ultrasonic treatment JP实验室股份有限公司 2026-05-19 CN claimed
WO-2026098831-A1 USE OF A PERSONAL CARE COMPOSITION FOR IMPROVING THE BARRIER FUNCTION OF SKIN UNILEVER IP HOLDINGS B.V. (NL) 2026-05-15 WO claimed
US-20260130837-A1 SPF BOOSTER AND SUNCARE FORMULATIONS INCLUDING SAME DOW SILICONES CORP (US) 2026-05-14 US claimed
CN-121566056-B Sulfonic modified ZIF-67 coated diaphragm and preparation method and application thereof 浙江理工大学 2026-05-12 CN claimed
WO-2026089857-A1 METHOD OF PREPARING AND USING A SKIN CARE COMPOSITION DOW SILICONES CORPORATION (US) 2026-04-30 WO claimed
WO-2026089856-A1 METHOD OF PREPARING AND USING A SKIN CARE FORMULATION DOW SILICONES CORPORATION (US) 2026-04-30 WO claimed
EP-4727519-A1 COSMETIC PREPARATION CONTAINING XANTHAN GUM AND VANILLIN DERIVATIVES Beiersdorf AG (DE) 2026-04-22 EP claimed
EP-4727521-A1 COSMETIC PREPARATION CONTAINING XANTHAN GUM AND ACETATES Beiersdorf AG (DE) 2026-04-22 EP claimed
EP-4727657-A1 COSMETIC PREPARATION CONTAINING XANTHAN GUM, TERPINENES AND TERPINEOL Beiersdorf AG (DE) 2026-04-22 EP claimed
US-20260102326-A1 SUNSCREEN COMPOSITION WITH LOW STICKINESS DSM IP ASSETS BV (NL) 2026-04-16 US claimed
US-4731242-A Waterproof sunscreen compositions PALINCZAR VICTOR (US) 1988-03-15 US claimed
US-4710371-A BUTENE POLYMER AND ULTRAVIOLET RADIATION ABSORBER PALINCZAR VICTOR (US) 1987-12-01 US claimed
US-4707354-A Mature skin treatment and protectant compositions and methods of using same ALPEN TAU, INC. (US) 1987-11-17 US claimed
US-4699779-A Waterproof sunscreen compositions PALINCZAR VICTOR 1987-10-13 US claimed
US-4686099-A Aerosol waterproof sunscreen compositions CHESEBROUGH-POND'S INC. 1987-08-11 US claimed
US-4683134-A HIGH VISCOSITY, GELS, ETHYL CELLULOSE, CROSSLINKED POLYACRYLIC ACID PALINCZAR VICTOR 1987-07-28 US claimed
US-4671956-A STABILITY; SIDE EFFECT REDUCTION L'OREAL (FR) 1987-06-09 US claimed
US-4671955-A ETHYL HYDROXYETHYL CELLULOSE AND AN ULTRAVIOLET RADIATION ABSORBER PALINCZAR VICTOR 1987-06-09 US claimed
US-4284621-A SUNSCREEN FOR SKIN BAYER AKTIENGESELLSCHAFT (DE) 1981-08-18 US claimed
EP-0005182-B1 COMPOSITION AGAINST THE ACTION OF LIGHT BAYER AG (DE) 1981-07-29 EP claimed