SCHEMBL3876046

SCHEMBL3876046

Cc1cc(-c2cc(N3CCN(c4ncccc4C(F)(F)F)CC3)nc(NS(=O)(=O)C(C)C)n2)ccc1F

nearest known ligand 0.43

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 10/20 0.43
GALR2 O43603 2/20 0.42
GALR1 P47211 2/20 0.42
TRPV1 Q8NER1 1/20 0.40
GAA P10253 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3948366 0.84 HSD11B1 (0.43) HSD11B1GALR2GALR1
SCHEMBL3878462 0.83 HSD11B1 (0.42) HSD11B1GALR2GALR1
SCHEMBL3884829 0.82 TRPV1 (0.46) HSD11B1GALR2GALR1TRPV1
SCHEMBL3880973 0.81 GALR2 (0.44) GALR2GALR1TRPV1GAA
SCHEMBL3877797 0.81 GALR2 (0.46) HSD11B1GALR2GALR1
SCHEMBL3888266 0.80 GALR2 (0.49) HSD11B1GALR2GALR1
SCHEMBL3877704 0.80 GALR2 (0.50) HSD11B1GALR2GALR1TRPV1
SCHEMBL3878777 0.80 GALR2 (0.43) HSD11B1GALR2GALR1TRPV1
SCHEMBL3887718 0.80 GAA (0.46) HSD11B1GALR2GALR1TRPV1GAA
SCHEMBL3881411 0.80 TRPV1 (0.45) GALR2GALR1TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7566712-B2 Biaryl piperazinyl-pyridine analogues NEUROGEN CORPORATION (US) 2009-07-28 US disclosed
US-7566712-B2 Biaryl piperazinyl-pyridine analogues NEUROGEN CORPORATION (US) 2009-07-28 US disclosed
US-7566712-B2 Biaryl piperazinyl-pyridine analogues NEUROGEN CORPORATION (US) 2009-07-28 US disclosed