SCHEMBL3877377

SCHEMBL3877377

Fc1ccc(-c2cc(N3CCN(c4ncccc4C(F)(F)F)CC3)nc(OCc3ccccc3C(F)(F)F)n2)cc1F

nearest known ligand 0.51

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
RBP4 P02753 1/20 0.46
HSD11B1 P28845 4/20 0.42
PIK3CA P42336 2/20 0.42
GALR2 O43603 2/20 0.40
GALR1 P47211 2/20 0.40
EPHX2 P34913 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3878855 0.81 GALR2 (0.48) HSD11B1GALR2GALR1EPHX2
SCHEMBL3877822 0.79 HSD11B1 (0.42) RBP4HSD11B1GALR2GALR1
SCHEMBL3884954 0.79 HSD11B1 (0.42) RBP4HSD11B1GALR2GALR1
SCHEMBL3880001 0.79 HSD11B1 (0.42) HSD11B1GALR2GALR1
SCHEMBL3877289 0.79 HSD11B1 (0.43) HSD11B1GALR2GALR1EPHX2
SCHEMBL3878811 0.79 GALR2 (0.46) RBP4HSD11B1GALR2GALR1
SCHEMBL3881034 0.78 MAPT (0.50) HSD11B1EPHX2
SCHEMBL3943144 0.78 HSD11B1 (0.42) HSD11B1GALR2GALR1
SCHEMBL3876557 0.78 GAA (0.47) RBP4HSD11B1GALR2GALR1
SCHEMBL3888965 0.78 GALR2 (0.49) PIK3CAGALR2GALR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7566712-B2 Biaryl piperazinyl-pyridine analogues NEUROGEN CORPORATION (US) 2009-07-28 US disclosed
US-7566712-B2 Biaryl piperazinyl-pyridine analogues NEUROGEN CORPORATION (US) 2009-07-28 US disclosed
US-7566712-B2 Biaryl piperazinyl-pyridine analogues NEUROGEN CORPORATION (US) 2009-07-28 US disclosed