SCHEMBL3879421

SCHEMBL3879421

CCN(CC)C1CCN(c2nc(-c3ccc(F)c(Cl)c3)cc(N3CCN(c4ncccc4C(F)(F)F)CC3)n2)CC1

nearest known ligand 0.45

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GALR2 O43603 4/20 0.45
GALR1 P47211 4/20 0.45
HSD11B1 P28845 7/20 0.40
TRPV1 Q8NER1 1/20 0.39
RBP4 P02753 1/20 0.38
MALT1 Q9UDY8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3882764 0.93 GALR2 (0.43) GALR2GALR1HSD11B1TRPV1
SCHEMBL3880207 0.89 GALR2 (0.51) GALR2GALR1HSD11B1TRPV1
SCHEMBL3876780 0.89 GALR2 (0.46) GALR2GALR1HSD11B1TRPV1RBP4
SCHEMBL3878568 0.88 TRPV1 (0.48) GALR2GALR1HSD11B1TRPV1RBP4
SCHEMBL3879455 0.88 GALR2 (0.46) GALR2GALR1HSD11B1TRPV1
SCHEMBL3880010 0.88 GALR2 (0.47) GALR2GALR1HSD11B1TRPV1
SCHEMBL3881028 0.87 GALR2 (0.44) GALR2GALR1HSD11B1TRPV1
SCHEMBL3877834 0.87 GALR2 (0.55) GALR2GALR1HSD11B1TRPV1
SCHEMBL3885408 0.87 GALR2 (0.55) GALR2GALR1HSD11B1TRPV1
SCHEMBL3888771 0.87 HSD11B1 (0.46) GALR2GALR1HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7566712-B2 Biaryl piperazinyl-pyridine analogues NEUROGEN CORPORATION (US) 2009-07-28 US disclosed
US-7566712-B2 Biaryl piperazinyl-pyridine analogues NEUROGEN CORPORATION (US) 2009-07-28 US disclosed
US-7566712-B2 Biaryl piperazinyl-pyridine analogues NEUROGEN CORPORATION (US) 2009-07-28 US disclosed