SCHEMBL3884795

SCHEMBL3884795

CNC(=O)c1cc(Oc2ccc3nc(NCCC4CCCCC4)oc3c2)ccn1

nearest known ligand 0.58

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
RAF1 P04049 15/20 0.58
BRAF P15056 15/20 0.58
KDR P35968 2/20 0.51
CSF1R P07333 4/20 0.50
PDGFRB P09619 1/20 0.50
KIT P10721 1/20 0.50
PDGFRA P16234 1/20 0.50
FLT3 P36888 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2677337 0.92 RAF1 (0.66) RAF1BRAFKDRCSF1RPDGFRB
SCHEMBL2675940 0.92 RAF1 (0.66) RAF1BRAFKDRCSF1RPDGFRB
SCHEMBL2677451 0.85 RAF1 (0.63) RAF1BRAFKDRCSF1RPDGFRB
SCHEMBL3884227 0.85 RAF1 (0.53) RAF1BRAFKDRCSF1RPDGFRB
SCHEMBL3884374 0.85 RAF1 (0.53) RAF1BRAFKDRCSF1RPDGFRB
SCHEMBL2676937 0.84 BRAF (0.53) RAF1BRAFKDRCSF1RKIT
SCHEMBL2675473 0.84 RAF1 (0.55) RAF1BRAFKDRCSF1RPDGFRB
SCHEMBL27738988 0.84 BRAF (0.62) RAF1BRAFKDR
SCHEMBL2676614 0.84 RAF1 (0.61) RAF1BRAFKDRCSF1RPDGFRB
SCHEMBL2676197 0.83 BRAF (0.54) RAF1BRAFKDRCSF1RKIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010528-A2 6-O-SUBSTITUTED BENZOXAZOLE AND BENZOTHIAZOLE COMPOUNDS AND METHODS OF INHIBITING CSF-1R SIGNALING Novartis Pharma AG (CH) 2009-01-07 EP claimed
WO-2007121484-A2 6-O-SUBSTITUTED BENZOXAZOLE AND BENZOTHIAZOLE COMPOUNDS AND METHODS OF INHIBITING CSF-1R SIGNALING NOVARTIS AG (CH) 2007-10-25 WO claimed