SCHEMBL3887740

SCHEMBL3887740

CC1CN(c2nccnc2Cl)CCN1c1cc(-c2ccc(F)c(F)c2)nc(Cl)n1

nearest known ligand 0.39

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 8/20 0.38
SMO Q99835 1/20 0.36
MALT1 Q9UDY8 1/20 0.35
KCNH2 Q12809 1/20 0.34
DGAT1 O75907 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13761506 1.00 TRPV1 (0.38) TRPV1SMOMALT1KCNH2DGAT1
SCHEMBL3879468 0.93 TRPV1 (0.38) TRPV1SMOMALT1
SCHEMBL13761549 0.93 MALT1 (0.40) TRPV1SMOMALT1
SCHEMBL3885538 0.93 MALT1 (0.40) TRPV1SMOMALT1
SCHEMBL3884028 0.93 MALT1 (0.40) TRPV1SMOMALT1
SCHEMBL3889401 0.92 TRPV1 (0.40) TRPV1SMOMALT1DGAT1
SCHEMBL3876436 0.92 SMO (0.41) TRPV1SMODGAT1
SCHEMBL3876440 0.92 SMO (0.41) TRPV1SMODGAT1
SCHEMBL3877069 0.89 TRPV1 (0.44) TRPV1
SCHEMBL3876588 0.89 TRPV1 (0.36) TRPV1MALT1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7566712-B2 Biaryl piperazinyl-pyridine analogues NEUROGEN CORPORATION (US) 2009-07-28 US disclosed