SCHEMBL3876440

SCHEMBL3876440

CC1CN(c2nccnc2Cl)CCN1c1cc(-c2ccc(F)cc2)nc(Cl)n1

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SMO Q99835 1/20 0.41
TRPV1 Q8NER1 9/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38
GSK3B P49841 1/20 0.38
MAPK1 P28482 1/20 0.35
HSD17B10 Q99714 1/20 0.35
DGAT1 O75907 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3876436 1.00 SMO (0.41) SMOTRPV1CYP1A2CYP2D6GSK3B
SCHEMBL13761506 0.92 TRPV1 (0.38) SMOTRPV1DGAT1
SCHEMBL3887740 0.92 TRPV1 (0.38) SMOTRPV1DGAT1
SCHEMBL3885538 0.91 MALT1 (0.40) SMOTRPV1
SCHEMBL3879468 0.91 TRPV1 (0.38) SMOTRPV1
SCHEMBL3884028 0.91 MALT1 (0.40) SMOTRPV1
SCHEMBL13761549 0.91 MALT1 (0.40) SMOTRPV1
SCHEMBL3889401 0.90 TRPV1 (0.40) SMOTRPV1DGAT1
SCHEMBL3991603 0.89 HSD17B10 (0.43) SMOTRPV1CYP1A2CYP2D6GSK3B
SCHEMBL13761561 0.88 SYK (0.41) SMOTRPV1CYP1A2CYP2D6GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7566712-B2 Biaryl piperazinyl-pyridine analogues NEUROGEN CORPORATION (US) 2009-07-28 US disclosed
US-20070027155-A1 Biaryl piperazinyl-pyridine analogues NEUROGEN CORPORATION 2007-02-01 US disclosed
CN-1823057-A Biaryl piperazinyl-pyridine analogues NEUROGEN CORP (US) 2006-08-23 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070027155-A1 Biaryl piperazinyl-pyridine analogues GPR174, GPR68, PPARG SMO 1465/4885TRPV1 244/4885CYP1A2 405/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.