SCHEMBL3892241

SCHEMBL3892241

CCCCCn1cc(Br)c(C#N)n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 5/20 0.39
MGAT2 Q10469 1/20 0.33
SMPD1 P17405 4/20 0.33
ALDH1A1 P00352 3/20 0.33
KDM4E B2RXH2 2/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CYP19A1 P11511 3/20 0.32
MAPK1 P28482 1/20 0.32
GLA P06280 1/20 0.32
POLB P06746 1/20 0.32
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32
HPGD P15428 1/20 0.32
CASP1 P29466 1/20 0.32
CASP7 P55210 1/20 0.32
HSD17B10 Q99714 1/20 0.32
SAE1 Q9UBE0 1/20 0.32
UBA2 Q9UBT2 1/20 0.32
TLR8 Q9NR97 1/20 0.31
TLR7 Q9NYK1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17066973 0.81 NPC1 (0.44) ALDH1A1KDM4ESMN1; SMN2MAPK1POLB
SCHEMBL2950186 0.76 L3MBTL1 (0.43) KDRSMPD1ALDH1A1KDM4ETLR8
SCHEMBL25413552 0.75 KDR (0.45) KDRSMPD1GBA1
SCHEMBL25415409 0.75 KDR (0.45) KDRSMPD1GBA1
SCHEMBL25415211 0.75 KDR (0.45) KDRSMPD1GBA1
SCHEMBL25414055 0.75 KDR (0.45) KDRSMPD1GBA1
SCHEMBL17943828 0.75 KDR (0.45) KDRSMPD1GBA1
SCHEMBL27592576 0.73 HSD17B10 (0.42) KDRALDH1A1MAPK1MAPTHPGD
SCHEMBL4374010 0.71
SCHEMBL2076920 0.71 KDR (0.49) KDRSMPD1ALDH1A1KDM4EGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2102170-A2 GLUCOCORTICOID MIMETICS, METHODS OF MAKING THEM, PHARMACEUTICAL COMPOSITIONS, AND USES THEREOF Boehringer Ingelheim International GmbH (DE) 2009-09-23 EP disclosed
WO-2008070507-A2 GLUCOCORTICOID MIMETICS, METHODS OF MAKING THEM, PHARMACEUTICAL COMPOSITIONS, AND USES THEREOF BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-06-12 WO disclosed