SCHEMBL3901003

SCHEMBL3901003

N#Cc1ccc(C(=O)N2CCC[C@@H]2COc2cccc(C#N)c2)cc1

nearest known ligand 0.63

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 3/20 0.59
HCRTR2 O43614 2/20 0.59
SPHK2 Q9NRA0 3/20 0.53
CPT1A P50416 1/20 0.46
DPP4 P27487 1/20 0.46
CHRNB4 P30926 2/20 0.45
CHRNA3 P32297 2/20 0.45
SPHK1 Q9NYA1 1/20 0.45
EGLN1 Q9GZT9 2/20 0.45
CHRNB2 P17787 1/20 0.45
CHRNA4 P43681 1/20 0.45
HRH3 Q9Y5N1 2/20 0.44
MGLL Q99685 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9240379 0.81 CHRNB4 (0.48) HCRTR1HCRTR2CHRNB4CHRNA3CHRNB2
SCHEMBL3912244 0.81 CHRNB4 (0.48) HCRTR1HCRTR2CHRNB4CHRNA3CHRNB2
SCHEMBL14132338 0.80 SPHK2 (0.53) HCRTR1HCRTR2SPHK2SPHK1
SCHEMBL3093335 0.80 HRH3 (0.53) HCRTR1HCRTR2DPP4HRH3
SCHEMBL3093346 0.80 HRH3 (0.53) HCRTR1HCRTR2DPP4HRH3
SCHEMBL3614551 0.78 CHRNB4 (0.69) CHRNB4CHRNA3CHRNB2CHRNA4
SCHEMBL9244259 0.78 CHRNB4 (0.69) CHRNB4CHRNA3CHRNB2CHRNA4
SCHEMBL4270669 0.77 HCRTR1 (0.55) HCRTR1HCRTR2SPHK2SPHK1EGLN1
SCHEMBL4270666 0.77 HCRTR1 (0.55) HCRTR1HCRTR2SPHK2SPHK1EGLN1
Hydrochloric Acid SCHEMBL9242770 0.77 CHRNB4 (0.67) CHRNB4CHRNA3CHRNB2CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0976722-B1 BENZAMIDINE DERIVATIVES AJINOMOTO KK (JP) 2009-03-11 EP disclosed
US-7396844-B1 Benzamidine derivatives AJINOMOTO CO., INC. (JP) 2008-07-08 US disclosed