SCHEMBL3902151

SCHEMBL3902151

Cc1ccc(C#N)cc1OCCN

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AR P10275 4/20 0.45
KDM4E B2RXH2 1/20 0.41
TRPV4 Q9HBA0 2/20 0.41
TSHR P16473 1/20 0.38
CYP19A1 P11511 1/20 0.38
CYP11B1 P15538 1/20 0.38
CYP11B2 P19099 1/20 0.38
ESR1 P03372 1/20 0.38
ICMT O60725 1/20 0.38
MAPT P10636 1/20 0.38
ALK Q9UM73 1/20 0.37
MRGPRX4 Q96LA9 1/20 0.37
TAAR1 Q96RJ0 1/20 0.37
LOXL2 Q9Y4K0 1/20 0.37
PTGDR2 Q9Y5Y4 1/20 0.37
ALDH1A1 P00352 1/20 0.36
CYP2A6 P11509 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25212014 0.88 MRGPRX4 (0.48) ARKDM4ETRPV4ESR1ICMT
SCHEMBL7356606 0.84 AR (0.46) ARKDM4ETRPV4TSHRCYP19A1
SCHEMBL27001716 0.83 AR (0.45) ARKDM4ETRPV4TSHRCYP19A1
SCHEMBL12460421 0.83 AR (0.49) ARKDM4ETRPV4TSHRCYP19A1
SCHEMBL13904208 0.81 KDM4E (0.40) ARKDM4ETRPV4CYP19A1CYP11B1
SCHEMBL3905446 0.81 KDM4E (0.40) ARKDM4ETRPV4CYP19A1CYP11B1
SCHEMBL5418640 0.80 TRPV4 (0.59) ARTRPV4MRGPRX4PTGDR2ALDH1A1
Hydrochloric Acid SCHEMBL3896102 0.80 KDM4E (0.43) ARKDM4ETRPV4CYP19A1CYP11B1
SCHEMBL12461366 0.80 MRGPRX4 (0.47) ARTRPV4ESR1ICMTMAPT
SCHEMBL25823520 0.78 TSHR (0.59) KDM4ETSHRTAAR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0976722-B1 BENZAMIDINE DERIVATIVES AJINOMOTO KK (JP) 2009-03-11 EP disclosed
US-7396844-B1 Benzamidine derivatives AJINOMOTO CO., INC. (JP) 2008-07-08 US disclosed
EP-0976722-A1 BENZAMIDINE DERIVATIVES Ajinomoto Co., Inc. (JP) 2000-02-02 EP disclosed
CN-1243505-A Benzamidine derivatives AJINOMOTO KK (JP) 2000-02-02 CN disclosed