SCHEMBL3909796

SCHEMBL3909796

Cc1cc(-c2nn(CC#N)cc2-c2ccnc(S(C)(=O)=O)n2)cc(O)c1C

nearest known ligand 0.45

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ROS1 P08922 12/20 0.45
ALK Q9UM73 9/20 0.39
MET P08581 1/20 0.39
BRAF P15056 5/20 0.35
TGFBR1 P36897 1/20 0.32
ALDH1A1 P00352 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14414410 0.87 BRAF (0.37) ROS1BRAFTGFBR1
SCHEMBL3918438 0.86 ROS1 (0.60) ROS1ALKMETBRAFTGFBR1
SCHEMBL3909956 0.85 ROS1 (0.41) ROS1ALKMETBRAF
SCHEMBL3979668 0.84 ROS1 (0.49) ROS1ALKMETBRAF
SCHEMBL3911878 0.84 ROS1 (0.49) ROS1ALKMETBRAF
SCHEMBL987733 0.81 ROS1 (0.54) ROS1ALKMETBRAF
SCHEMBL3911292 0.81 ROS1 (0.51) ROS1ALKMETBRAF
SCHEMBL3911285 0.81 ROS1 (0.51) ROS1ALKMETBRAF
SCHEMBL3911904 0.79 ROS1 (0.45) ROS1ALKMETBRAF
SCHEMBL3918762 0.79 ROS1 (0.44) ROS1ALKMETBRAFALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2024353-A2 PYRAZOLE COMPOUNDS Pfizer Products Inc. (US) 2009-02-18 EP disclosed
WO-2007105058-A2 PYRAZOLE COMPOUNDS PFIZER PRODUCTS INC. (US) 2007-09-20 WO disclosed