SCHEMBL3979668

SCHEMBL3979668

CS(=O)(=O)c1nccc(-c2cn(CC#N)nc2-c2cc(O)cc(Cl)c2)n1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ROS1 P08922 10/20 0.49
ALK Q9UM73 7/20 0.43
MET P08581 1/20 0.43
BRAF P15056 8/20 0.40
MAPK14 Q16539 2/20 0.34
PTGS2 P35354 1/20 0.32
MAP4K4 O95819 1/20 0.32
EGFR P00533 1/20 0.32
FRK P42685 1/20 0.32
MAPK9 P45984 1/20 0.32
CSNK1D P48730 1/20 0.32
SLK Q9H2G2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3918438 0.91 ROS1 (0.60) ROS1ALKMETBRAF
SCHEMBL3911878 0.90 ROS1 (0.49) ROS1ALKMETBRAFPTGS2
SCHEMBL3911904 0.87 ROS1 (0.45) ROS1ALKMETBRAFMAPK14
SCHEMBL3909956 0.86 ROS1 (0.41) ROS1ALKMETBRAFMAPK14
SCHEMBL3909796 0.84 ROS1 (0.45) ROS1ALKMETBRAF
SCHEMBL1557302 0.84 ROS1 (0.49) ROS1ALKMETBRAF
SCHEMBL14414507 0.83 ROS1 (0.49) ROS1ALKMETBRAFMAPK14
SCHEMBL3908117 0.82 ROS1 (0.50) ROS1ALKMETBRAF
SCHEMBL3912171 0.81 ROS1 (0.37) ROS1ALKBRAFMAPK14MAPK9
SCHEMBL3912514 0.80 ROS1 (0.55) ROS1ALKMETBRAFMAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2024353-A2 PYRAZOLE COMPOUNDS Pfizer Products Inc. (US) 2009-02-18 EP disclosed
WO-2007105058-A2 PYRAZOLE COMPOUNDS PFIZER PRODUCTS INC. (US) 2007-09-20 WO disclosed
WO-2007105058-A2 PYRAZOLE COMPOUNDS PFIZER PRODUCTS INC. (US) 2007-09-20 WO disclosed