SCHEMBL3910012

SCHEMBL3910012

CO[Si](C)(CCCCNC(N)=O)OC

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 5/20 0.37
KDM4E B2RXH2 1/20 0.35
MAPK1 P28482 1/20 0.35
HIF1A Q16665 1/20 0.35
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
PAOX Q6QHF9 2/20 0.34
MTNR1A P48039 2/20 0.33
MTNR1B P49286 2/20 0.33
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33
TSHR P16473 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA9 Q16790 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3912407 0.98 EPHX1 (0.40) EPHX1KDM4EMAPK1HIF1AMEN1
SCHEMBL3907811 0.98 EPHX1 (0.40) EPHX1KDM4EMAPK1HIF1AMEN1
SCHEMBL3916905 0.98 EPHX1 (0.40) EPHX1KDM4EMAPK1HIF1AMEN1
SCHEMBL3909839 0.98 EPHX1 (0.40) EPHX1KDM4EMAPK1HIF1AMEN1
SCHEMBL3916972 0.98 EPHX1 (0.40) EPHX1KDM4EMAPK1HIF1AMEN1
SCHEMBL3918921 0.98 EPHX1 (0.40) EPHX1KDM4EMAPK1HIF1AMEN1
SCHEMBL3912112 0.98 EPHX1 (0.40) EPHX1KDM4EMAPK1HIF1AMEN1
SCHEMBL3913334 0.98 EPHX1 (0.40) EPHX1KDM4EMAPK1HIF1AMEN1
SCHEMBL114474 0.94 EPHX1 (0.34) EPHX1KDM4EMAPK1HIF1AMEN1
SCHEMBL3917119 0.86 MTNR1A (0.35) MTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090277559-A1 METHOD FOR VULCANIZATION-ADHERING RUBBER COMPOSITION TO ADHERENT OF BRASS OR PLATED WITH BRASS, REINFORCING MEMBER FOR RUBBER ARTICLE, RUBBER-REINFORCING MEMBER COMPOSITE AND PNEUMATIC TIRE BRIDGESTONE CORPORATION (JP) 2009-11-12 US disclosed
EP-1840158-B1 METHOD FOR VULCANIZATION AND ADHESION OF RUBBER COMPOSITION WITH ARTICLE TO BE ADHERED BEING MADE OF BRASS OR PLATED WITH BRASS, REINFORCING MATERIAL FOR RUBBER ARTICLE, RUBBER-REINFORCING MATERIAL COMPOSITE, AND PNEUMATIC TIRE BRIDGESTONE CORP (JP) 2009-02-18 EP disclosed
EP-1840158-A1 METHOD FOR VULCANIZATION AND ADHESION OF RUBBER COMPOSITION WITH ARTICLE TO BE ADHERED BEING MADE OF BRASS OR PLATED WITH BRASS, REINFORCING MATERIAL FOR RUBBER ARTICLE, RUBBER-REINFORCING MATERIAL COMPOSITE, AND PNEUMATIC TIRE Bridgestone Corporation (JP) 2007-10-03 EP disclosed