SCHEMBL3918944

SCHEMBL3918944

CC#CCn1c(Br)nc2c1c(=O)n(Cc1ncc(C#N)c3ccccc13)c(=O)n2C

nearest known ligand 0.54

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 19/20 0.54
KCNH2 Q12809 4/20 0.46
CHRM1 P11229 1/20 0.45
KMT2A Q03164 1/20 0.43
FAP Q12884 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL497449 0.84 DPP4 (0.50) DPP4KCNH2KMT2A
SCHEMBL9290262 0.83 DPP4 (0.51) DPP4KCNH2CHRM1FAP
SCHEMBL3919809 0.83 DPP4 (0.68) DPP4KCNH2FAP
SCHEMBL638215 0.83 DPP4 (0.55) DPP4KCNH2CHRM1FAP
SCHEMBL4487837 0.83 KMT2A (0.60) DPP4KMT2A
SCHEMBL3918551 0.82 DPP4 (0.51) DPP4CHRM1FAP
SCHEMBL9290265 0.82 DPP4 (0.49) DPP4KCNH2CHRM1FAP
SCHEMBL8273211 0.82 DPP4 (0.49) DPP4KCNH2CHRM1FAP
SCHEMBL3975825 0.80 DPP4 (0.84) DPP4CHRM1FAP
SCHEMBL3975831 0.80 DPP4 (0.84) DPP4CHRM1FAP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7550455-B2 8-(piperazin-1yl)- and 8-([1,4]diazepan-1yl)-xanthines, the preparation thereof and their use as pharmaceutical composition BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-06-23 US disclosed