SCHEMBL9290262

SCHEMBL9290262

CC#CCn1c(N(C)CCN)nc2c1c(=O)n(Cc1ncc(C#N)c3ccccc13)c(=O)n2C

nearest known ligand 0.51

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 20/20 0.51
KCNH2 Q12809 3/20 0.43
CHRM1 P11229 1/20 0.42
FAP Q12884 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8273223 0.90 DPP4 (0.51) DPP4KCNH2CHRM1FAP
SCHEMBL8273211 0.89 DPP4 (0.49) DPP4KCNH2CHRM1FAP
SCHEMBL9290265 0.89 DPP4 (0.49) DPP4KCNH2CHRM1FAP
SCHEMBL13936198 0.88 DPP4 (0.55) DPP4KCNH2CHRM1FAP
SCHEMBL8272361 0.87 DPP4 (0.61) DPP4CHRM1FAP
SCHEMBL13936184 0.86 DPP4 (0.47) DPP4KCNH2CHRM1FAP
SCHEMBL8272025 0.86 DPP4 (0.47) DPP4KCNH2CHRM1FAP
SCHEMBL13936187 0.85 KMT2A (0.53) DPP4
SCHEMBL8273232 0.85 DPP4 (0.46) DPP4CHRM1FAP
SCHEMBL3918944 0.83 DPP4 (0.54) DPP4KCNH2CHRM1FAP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1797093-B1 NOVEL 3-METHYL-7-BUTINYL-XANTHINES, PRODUCTION THEREOF, AND USE THEREOF AS MEDICAMENTS BOEHRINGER INGELHEIM INT (DE) 2012-05-30 EP disclosed
US-7495002-B2 3-methyl-7-butinyl-xanthines, the preparation thereof and their use as pharmaceutical compositions BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-02-24 US disclosed
US-7495002-B2 3-methyl-7-butinyl-xanthines, the preparation thereof and their use as pharmaceutical compositions BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-02-24 US disclosed