SCHEMBL3919981

SCHEMBL3919981

CS(=O)(=O)N1CCN(Cc2ccc(C(N)=O)cc2C(F)(F)F)CC1

nearest known ligand 0.62

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.62
ALDH1A1 P00352 7/20 0.50
KDM4E B2RXH2 6/20 0.50
NR1H2 P55055 1/20 0.48
DDR1 Q08345 6/20 0.46
TDP1 Q9NUW8 4/20 0.46
RECQL P46063 1/20 0.46
GAA P10253 2/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
KIT P10721 2/20 0.44
HPGD P15428 1/20 0.43
ATM Q13315 1/20 0.43
ALOX15 P16050 2/20 0.42
HTT P42858 1/20 0.42
MAPT P10636 1/20 0.42
BRAF P15056 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31536436 0.87 NR1H2 (0.59) NR1H2DDR1KITBRAF
SCHEMBL3311056 0.85 NR1H2 (0.52) NR1H2DDR1KITATMHTT
SCHEMBL2707620 0.85 NR1H2 (0.66) ALDH1A1KDM4ENR1H2DDR1KIT
SCHEMBL2777362 0.84 DDR1 (0.51) NPSR1ALDH1A1KDM4ENR1H2DDR1
SCHEMBL30899974 0.83 NPSR1 (0.59) NPSR1ALDH1A1KDM4EKITBRAF
SCHEMBL3919971 0.83 NR1H2 (0.70) NPSR1ALDH1A1KDM4ENR1H2DDR1
SCHEMBL16380735 0.83 NR1H2 (0.49) NPSR1ALDH1A1KDM4ENR1H2DDR1
SCHEMBL16380700 0.83 DDR1 (0.50) NPSR1ALDH1A1KDM4ENR1H2DDR1
SCHEMBL2707798 0.82 DDR1 (0.56) NPSR1ALDH1A1KDM4ENR1H2DDR1
SCHEMBL3992921 0.82 IP6K1 (0.52) NPSR1ALDH1A1KDM4EDDR1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2038253-A1 BIPHENYL DERIVATIVES AND THEIR USE IN TREATING HEPATITIS C Arrow Therapeutics Limited (GB) 2009-03-25 EP disclosed
WO-2007138242-A1 BIPHENYL DERIVATIVES AND THEIR USE IN TREATING HEPATITIS C ARROW THERAPEUTICS LIMITED (GB) 2007-12-06 WO disclosed