SCHEMBL3920104

SCHEMBL3920104

CCCCc1cccc(N=C=O)c1C

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.59
GABRA1 P14867 2/20 0.47
GABRB2 P47870 2/20 0.47
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
BID P55957 3/20 0.35
MCL1 Q07820 3/20 0.35
BCL2L1 Q07817 2/20 0.35
BAK1 Q16611 2/20 0.35
KAT8 Q9H7Z6 2/20 0.35
PPARA Q07869 2/20 0.35
PPARG P37231 1/20 0.35
EP300 Q09472 1/20 0.35
KAT2A Q92830 1/20 0.35
KAT2B Q92831 1/20 0.35
KAT5 Q92993 1/20 0.35
SAE1 Q9UBE0 1/20 0.35
TRPA1 O75762 1/20 0.34
LIPG Q9Y5X9 1/20 0.33
ALOX5 P09917 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2346860 0.87 CYP3A4 (0.50) CYP3A4GABRA1GABRB2CYP2D6CYP2C9
SCHEMBL993745 0.85 CYP3A4 (0.51) CYP3A4GABRA1GABRB2CYP2D6CYP2C9
SCHEMBL29651833 0.85 CYP3A4 (0.51) CYP3A4GABRA1GABRB2CYP2D6CYP2C9
SCHEMBL23522251 0.84 CYP3A4 (0.70) CYP3A4GABRA1GABRB2TRPA1
SCHEMBL1551949 0.83 CYP3A4 (0.57) CYP3A4GABRA1GABRB2CYP2D6CYP2C9
SCHEMBL10965705 0.82 CYP3A4 (0.45) CYP3A4GABRA1GABRB2CYP2D6CYP2C9
SCHEMBL6419136 0.81 CYP3A4 (0.70) CYP3A4GABRA1GABRB2TRPA1
SCHEMBL10971614 0.80 CYP3A4 (0.46) CYP3A4GABRA1GABRB2CYP2D6CYP2C9
SCHEMBL2350176 0.80 CYP3A4 (0.46) CYP3A4GABRA1GABRB2CYP2D6CYP2C9
SCHEMBL17847485 0.79 CYP3A4 (0.43) CYP3A4GABRA1GABRB2CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009003669-A2 PYRIDO(3,2-D)PYRIMIDINES AND PHARMACEUTICAL COMPOSITIONS USEFUL FOR MEDICAL TREATMENT 4 AZA IP NV (BE) 2009-01-08 WO disclosed