SCHEMBL3924176

SCHEMBL3924176

O=[N+]([O-])c1cc(OCc2ccccc2)c(OCc2ccccc2)c(-c2nc(-c3cccnc3C(F)(F)F)no2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 4/20 0.43
CYP11B1 P15538 2/20 0.43
CYP11B2 P19099 2/20 0.43
MAPT P10636 5/20 0.40
GAA P10253 2/20 0.38
POLB P06746 1/20 0.38
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
NPC1 O15118 3/20 0.38
RXFP1 Q9HBX9 1/20 0.38
PPIA P62937 2/20 0.38
TDP1 Q9NUW8 1/20 0.37
PPIF P30405 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
HDAC5 Q9UQL6 1/20 0.37
PTGES O14684 1/20 0.37
RAB9A P51151 2/20 0.37
GRM5 P41594 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3581595 0.85 POLB (0.47) MAPTPOLBNPC1RXFP1RAB9A
SCHEMBL1447240 0.84 POLB (0.46) MAPTPOLBNPC1RXFP1RAB9A
SCHEMBL9388459 0.71 MEN1 (0.58) CYP19A1CYP11B1CYP11B2MAPTMEN1
SCHEMBL3590056 0.71 EIF4E (0.44) CYP19A1CYP11B1CYP11B2MEN1KMT2A
SCHEMBL1447215 0.71 POLB (0.43) MAPTGAAPOLBNPC1RXFP1
SCHEMBL1447848 0.68 POLB (0.42) MAPTPOLBNPC1RXFP1RAB9A
SCHEMBL3581708 0.68 TUBB4A (0.41) CYP19A1CYP11B1CYP11B2MEN1KMT2A
SCHEMBL5865429 0.68 MAPT (0.71) CYP19A1CYP11B1CYP11B2MAPTGAA
SCHEMBL3587958 0.68 PPIA (0.41) CYP19A1CYP11B1CYP11B2MAPTMEN1
SCHEMBL8077523 0.67 CYP19A1 (0.55) CYP19A1CYP11B1CYP11B2MAPTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2027091-A1 NEW PHARMACEUTICAL COMPOUNDS BIAL - Portela & Ca., S.A. (PT) 2009-02-25 EP disclosed
WO-2007117165-A1 NEW PHARMACEUTICAL COMPOUNDS BIAL - PORTELA & CA, S.A. (PT) 2007-10-18 WO disclosed