SCHEMBL3925943

SCHEMBL3925943

CC(C)(C)OC(=O)N1CCC(COCCc2cc(Br)cc3nccnc23)(c2ccc(F)cc2)CC1

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 10/20 0.46
SLC6A4 P31645 8/20 0.39
KCNH2 Q12809 8/20 0.39
RORC P51449 5/20 0.37
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35
GRIA1 P42261 1/20 0.35
OPRD1 P41143 1/20 0.35
OPRK1 P41145 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3924571 0.89 TACR1 (0.44) TACR1SLC6A4KCNH2RORCHDAC1
SCHEMBL3925962 0.88 TACR1 (0.44) TACR1SLC6A4KCNH2RORC
SCHEMBL3935051 0.85 TACR1 (0.51) TACR1SLC6A4KCNH2
SCHEMBL4204373 0.83 TACR1 (0.42) TACR1RORCHDAC1HDAC2OPRD1
SCHEMBL4305041 0.80 TACR1 (0.47) TACR1SLC6A4KCNH2RORCGRIA1
SCHEMBL4291217 0.79 TACR1 (0.43) TACR1SLC6A4KCNH2RORC
SCHEMBL4027722 0.77 TACR1 (0.55) TACR1SLC6A4KCNH2
SCHEMBL3921939 0.77 TACR1 (0.43) TACR1SLC6A4KCNH2RORCHDAC1
SCHEMBL3934912 0.76 TACR1 (0.42) TACR1SLC6A4KCNH2RORCHDAC1
SCHEMBL3928337 0.75 TACR1 (0.51) TACR1SLC6A4KCNH2RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009009633-A1 SUBSTITUTED HETEROCYCLIC ETHERS AND THEIR USE IN CNS DISORDERS BRISTOL-MYERS SQUIBB COMPANY (US) 2009-01-15 WO disclosed