SCHEMBL4305041

SCHEMBL4305041

CC(C)(C)OC(=O)N1CCC(COCCc2ccc(C(F)(F)F)c3cccnc23)(c2ccc(F)cc2)CC1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 6/20 0.47
RORC P51449 5/20 0.39
SLC6A4 P31645 2/20 0.39
KCNH2 Q12809 2/20 0.39
OPRD1 P41143 1/20 0.38
OPRK1 P41145 1/20 0.38
DTYMK P23919 1/20 0.38
EPHX2 P34913 1/20 0.37
POLB P06746 1/20 0.36
SQOR Q9Y6N5 1/20 0.35
CCR5 P51681 1/20 0.35
GRIA1 P42261 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4207977 0.82 TACR1 (0.43) TACR1RORCSLC6A4KCNH2OPRD1
SCHEMBL3924571 0.82 TACR1 (0.44) TACR1RORCSLC6A4KCNH2OPRD1
SCHEMBL4291217 0.80 TACR1 (0.43) TACR1RORCSLC6A4KCNH2SQOR
SCHEMBL3925943 0.80 TACR1 (0.46) TACR1RORCSLC6A4KCNH2OPRD1
SCHEMBL3925962 0.78 TACR1 (0.44) TACR1RORCSLC6A4KCNH2
SCHEMBL18280071 0.75 GPR119 (0.47) DTYMKEPHX2POLB
SCHEMBL3928378 0.75 TACR1 (0.53) TACR1RORCSLC6A4KCNH2
SCHEMBL3565915 0.73 POLB (0.50) DTYMKPOLB
SCHEMBL4027722 0.73 TACR1 (0.55) TACR1SLC6A4KCNH2
SCHEMBL3921939 0.73 TACR1 (0.43) TACR1RORCSLC6A4KCNH2CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009009633-A1 SUBSTITUTED HETEROCYCLIC ETHERS AND THEIR USE IN CNS DISORDERS BRISTOL-MYERS SQUIBB COMPANY (US) 2009-01-15 WO disclosed